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Search Count: 6

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5I5Z image
Cdk8-Cycc In Complex With 8-(1-Methyl-2,2-Dioxo-2,3-Dihydro-1H-2L6-Benzo[C]Isothiazol-5-Yl)-[1,6]Naphthyridine-2-Carboxylic Acid Methylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2016-04-13
Classification: TRANSFERASE
Ligands: 68U, FMT

5FGK image
Cdk8-Cycc In Complex With 8-[3-(3-Amino-1H-Indazol-6-Yl)-5-Chloro- Pyridine-4-Yl]-2,8-Diaza-Spiro[4.5]Decan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.36 Å Release Date: 2016-02-03
Classification: TRANSFERASE
Ligands: 5XG, DMS, EDO, FMT

5HBE image
Cdk8-Cycc In Complex With 8-[3-Chloro-5-(1-Methyl-2,2-Dioxo-2, 3-Dihydro-1H-2L6-Benzo[C]Isothiazol-5-Yl)-Pyridin- 4-Yl]-1-Oxa-3,8-Diaza-Spiro[4.5]Decan-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.38 Å Release Date: 2016-02-03
Classification: TRANSFERASE
Ligands: 5Y6, DMS, EDO, FMT

5HBH image
Cdk8-Cycc In Complex With 5-{5-Chloro-4-[1-(2-Methoxy-Ethyl)-1,8-Diaza-Spiro[4.5]Dec-8-Yl]-Pyridin-3-Yl}-1-Methyl-1,3-Dihydro-Benzo[C]Isothiazole 2,2-Dioxide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2016-02-03
Classification: TRANSFERASE
Ligands: 5Y7, EDO, FMT

5HBJ image
Cdk8-Cycc In Complex With 8-[2-Amino-3-Chloro-5-(1-Methyl-1H-Indazol-5-Yl)-Pyridin-4-Yl]-2,8-Diaza-Spiro[4.5]Decan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2016-02-03
Classification: TRANSFERASE
Ligands: 5Y8, EDO, FMT

5BNJ image
Cdk8/Cycc In Complex With 8-{3-Chloro-5-[4-(1-Methyl-1H-Pyrazol-4-Yl)-Phenyl]-Pyridin- 4-Yl}-2,8-Diaza-Spiro[4.5]Decan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.64 Å Release Date: 2015-10-14
Classification: TRANSFERASE
Ligands: 4TV, FMT
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