Search Count: 20
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2019-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: Z3A
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Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 9EM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 9EM
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 9J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 9J4
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2014-12-24 Classification: TRANSFERASE/INHIBITOR Ligands: 3QX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3QX
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Crystal Structure Of Mitogen-Activated Protein Kinase 14 (P38-H5) Complex With 5-(2-Chlorophenyl)-N-(5-(Cyclopropylcarbamoyl)-2-Methylphenyl)-2-Thiophenecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2013-06-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1M8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-12
Ligands: 1M8
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Crystal Structure Of Mitogen-Activated Protein Kinase 14 (P38-H5) Complex With 2-(2-Chlorophenyl)-N-(5-(Cyclopropylcarbamoyl)-2-Methylphenyl)-1,3-Thiazole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2013-06-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1R9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-12
Ligands: 1R9
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Crystal Structure Of Mitogen-Activated Protein Kinase 14 (P38-H5) Complex With Ethyl 6-((5-(Cyclopropylcarbamoyl)-2-Methylphenyl)Carbamoyl)-1H-Indole-1-Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-06-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1RA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-12
Ligands: 1RA
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P38 Alpha Kinase Complexed With A Pyrazolo-Triazine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: NK0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: NK0
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P38 Alpha Kinase Complexed With A 5-Amino-Pyrazole Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2010-11-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OCG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-17
Ligands: OCG
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: 38P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 38P
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7V
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-10-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 39P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 39P
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P38 Alpha Kinase Complexed With A 2-Aminothiazol-5-Yl-Pyrimidine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2010-09-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3NW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: 3NW
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P38 Alpha Kinase Complexed With A Pyrazolo-Pyrimidine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-03-02 Classification: TRANSFERASE Ligands: N4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: N4D
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Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2008-04-15 Classification: TRANSFERASE Ligands: P39 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: P39
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P38 Alpha Map Kinase Complexed With Bms-640994
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-15 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: 304 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: 304
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Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-08 Classification: TRANSFERASE Ligands: P38 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
Ligands: P38
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P38 Alpha Map Kinase Complexed With A Benzothiazole Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2008-03-25 Classification: TRANSFERASE Ligands: P41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-25
Ligands: P41
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 279 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 279
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Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 287 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 287
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P38 Alpha Map Kinase Inhibitor Based On Heterobicyclic Scaffolds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2007-08-21 Classification: TRANSFERASE Ligands: LGF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-21
Ligands: LGF
