Search Count: 17
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Crystal Structure Of The Mertk Kinase Domain With Sa4488
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-10-09 Classification: TRANSFERASE Ligands: A1APF, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APF, CL
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Mertk In Complex With Small Molecule 6-{1-[([1,1'-Biphenyl]-4-Yl)Carbamoyl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APG, CL
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Mertk In Complex With Small Molecule Inhibitor 6-{1-[6-(3-Hydroxy-3-Methylbutoxy)-1,3-Benzoxazol-2-Yl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APH, CL
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Cdk2 With Compound 14 Inhibitor With Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-07-07 Classification: SIGNALING PROTEIN, Transferase/Inhibitor Ligands: YOS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: YOS
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Gsk-3Beta With Inhibitor 6-Chloro-N-Cyclohexyl-4-(1H-Pyrrolo[2,3-B]Pyridin-3-Yl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.12 Å Release Date: 2013-04-24 Classification: Transferase/Transferase Inhibitor Ligands: IQ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: IQ6
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Parp Complexed With A906894
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-12-22 Classification: Transferase/Transferase Inhibitor Ligands: L3L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: L3L
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Parp Complexed With A927929
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-06-23 Classification: TRANSFERASE Ligands: A92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-23
Ligands: A92
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Parp Complexed With A968427
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-03-09 Classification: TRANSFERASE Ligands: GJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: GJW
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Pka Structures Of Akt, Indazole-Pyridine Inhibitors
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-06-05 Classification: TRANSFERASE Ligands: SS3 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: SS3
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Pka Structures Of Indazole-Pyridine Series Of Akt Inhibitors
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-06-05 Classification: TRANSFERASE Ligands: L20 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: L20
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Pka Structures Of Indazole-Pyridine Series Of Akt Inhibitors
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-06-05 Classification: TRANSFERASE Ligands: SS5 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: SS5
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Pka Structures Of Indazole-Pyridine Series Of Akt Inhibitors
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-06-05 Classification: TRANSFERASE Ligands: SS4 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2007-06-05
Ligands: SS4
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Cyclooxygenase-2 (Prostaglandin Synthase-2) Complexed With A Selective Inhibitor, Sc-558
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 1997-12-24 Classification: OXIDOREDUCTASE Ligands: NAG, HEM, S58 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1997-12-24
Ligands: NAG, HEM, S58
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Cyclooxygenase-2 (Prostaglandin Synthase-2) Complexed With A Non-Selective Inhibitor, Flurbiprofen
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1997-12-24 Classification: OXIDOREDUCTASE Ligands: NAG, HEM, FLP |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1997-12-24
Ligands: NAG, HEM, FLP
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Cyclooxygenase-2 (Prostaglandin Synthase-2) Complexed With A Non-Selective Inhibitor, Indomethacin
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 1997-12-24 Classification: OXIDOREDUCTASE Ligands: NAG, HEM, IMN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1997-12-24
Ligands: NAG, HEM, IMN
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Uninhibited Mouse Cyclooxygenase-2 (Prostaglandin Synthase-2)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 1997-12-24 Classification: OXIDOREDUCTASE Ligands: NAG, HEM |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1997-12-24
Ligands: NAG, HEM
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Cyclooxygenase-2 (Prostaglandin Synthase-2) Complexed With A Selective Inhibitor, Sc-558 In I222 Space Group
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 1997-12-24 Classification: OXIDOREDUCTASE Ligands: NAG, HEM, S58 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1997-12-24
Ligands: NAG, HEM, S58
