Search Count: 17
![]() |
Rho-Associated Protein Kinase 1 (Rock 1) In Complex With Rki1447
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2012-08-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 07R, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-22
Ligands: 07R, EDO
![]() |
Human Rho-Associated Protein Kinase 1 (Rock 1) In Complex With Indazole Derivative (Compound 18)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2012-02-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0HD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: 0HD
![]() |
Crystal Structure Of Hcv Ns5B Polymerase With A Novel Monocyclic Dihydropyridinone Inhibitor
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2009-12-08 Classification: TRANSFERASE Ligands: B42 |
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION
Release Date: 2009-12-08
Ligands: B42
![]() |
Crystal Structure Of Hcv Ns5B Polymerase In Complex With A Novel Bicyclic Dihydro-Pyridinone Inhibitor
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-12-08 Classification: TRANSFERASE Ligands: YAK |
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION
Release Date: 2009-12-08
Ligands: YAK
![]() |
Crystal Structure Of Hcv Ns5B Polymerase With A Novel Monocyclic Dihydro-Pyridinone Inhibitor
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-12-08 Classification: TRANSFERASE Ligands: B80 |
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION
Release Date: 2009-12-08
Ligands: B80
![]() |
Crystal Structure Of Hcv Ns5B Polymerase With A Novel Pyridazinone Inhibitor
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-08-18 Classification: TRANSFERASE Ligands: N35 |
Organism: Hepatitis c virus (isolate bk)
Method: X-RAY DIFFRACTION
Release Date: 2009-08-18
Ligands: N35
![]() |
The Structure Of Dpp4 In Complex With Piperidine Fused Benzimidazole 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-07-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, NA, 677 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-21
Ligands: NAG, NA, 677
![]() |
The Structure Of Dpp-4 In Complex With Piperidine Fused Imidazopyridine 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-07-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, NA, 361 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-21
Ligands: NAG, NA, 361
![]() |
Human Dipeptidyl Peptidase Iv/Cd26 In Complex With A Flouroolefin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-04-22 Classification: HYDROLASE Ligands: NAG, 315 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: NAG, 315
![]() |
Human Dipeptidyl Peptidase Iv/Cd26 In Complex With A Fluoroolefin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2008-04-22 Classification: HYDROLASE Ligands: NAG, NA, 317 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: NAG, NA, 317
![]() |
Human Dipeptidyl Peptidase Iv In Complex With A Triazolopiperazine-Based Beta Amino Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: NAG, NA, 448 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: NAG, NA, 448
![]() |
Human Dipeptidyl Peptidase Iv/Cd26 In Complex With A 4-Aryl Cyclohexylalanine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: NAG, NA, 524 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: NAG, NA, 524
![]() |
Human Dipeptidyl Peptidase Iv/Cd26 In Complex With A 4-Aryl Cyclohexylalanine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: NAG, NA, 474 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: NAG, NA, 474
![]() |
Human Dipeptidyl Peptidase Iv In Complex With An Alpha Amino Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-05-08 Classification: HYDROLASE Ligands: NAG, NA, 277 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-05-08
Ligands: NAG, NA, 277
![]() |
The Structure Of Dpp4 In Complex With An Oxadiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2006-09-19 Classification: HYDROLASE Ligands: NAG, NA, 3TP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-19
Ligands: NAG, NA, 3TP
![]() |
Human Dipeptidyl Peptidase Iv/Cd26 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2006-07-04 Classification: HYDROLASE Ligands: NAG, S14 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-07-04
Ligands: NAG, S14
![]() |
Human Dipeptidyl Peptidase Iv In Complex With A Beta Amino Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2005-01-18 Classification: HYDROLASE Ligands: NAG, NA, 715 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-18
Ligands: NAG, NA, 715
