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9NWS image
Cryo-Em Structure Of Ddb1Db:Crbn:Mezigdomide:Sall4(392-449)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-02-04
Classification: LIGASE
Ligands: ZN, QFC

9NWT image
Cryo-Em Structure Of Ddb1Db:Crbn:Mezigdomide:Sall4(392-449;G416A)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-02-04
Classification: LIGASE
Ligands: ZN, QFC

9Q22 image
Crystal Structure Of Ternary Complex Helios-Zf2:I-19:Crbn:Ddb1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.41 Å Release Date: 2025-10-01
Classification: LIGASE
Ligands: A1CNP, ZN

9Q2D image
Cryo-Em Structure Of Ternary Complex Ikaros-Zf2:Cc-885:Crbn:Ddb1 (Molecular Glue Degrader)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Resolution:2.94 Å Release Date: 2025-10-01
Classification: LIGASE
Ligands: ZN, 85C

9E2U image
Crystal Structure Of Ddb1-Crbn-Alv1 Complex Bound To Triple Znf Of Helios (Ikzf2 Zf1-3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:4.11 Å Release Date: 2025-09-03
Classification: LIGASE
Ligands: RN9, ZN

9B9R image
Cryo-Em Structure Of The Zbtb5 Btb Domain Filament
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-07-24
Classification: TRANSCRIPTION

9B9V image
Cryo-Em Structure Of The Zbtb9 Btb Domain Filament
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-07-24
Classification: TRANSCRIPTION

8P82 image
Cryo-Em Structure Of Dimeric Ubr5
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-06-14
Classification: LIGASE
Ligands: ZN

8P83 image
Cryo-Em Structure Of Full-Length Human Ubr5 (Homotetramer)
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-06-14
Classification: LIGASE

8G46 image
Cryo-Em Structure Of Ddb1Deltab-Dda1-Dcaf16-Brd4(Bd2)-Mmh2
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Resolution:2.20 Å Release Date: 2023-03-08
Classification: LIGASE
Ligands: ZN, YK3

7KXD image
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.62 Å Release Date: 2021-01-20
Classification: TRANSFERASE/Agonist
Ligands: Z7G

7KXE image
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.42 Å Release Date: 2021-01-20
Classification: TRANSFERASE/Agonist
Ligands: Z7H

7KXF image
Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.14 Å Release Date: 2021-01-20
Classification: TRANSFERASE/Agonist
Ligands: Z7I

6CJ2 image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg056
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.47 Å Release Date: 2019-03-06
Classification: TRANSCRIPTION/INHIBITOR
Ligands: X27

6CD5 image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Xmd17-26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.58 Å Release Date: 2019-01-16
Classification: TRANSCRIPTION/INHIBITOR
Ligands: R4L, EDO, NO3

6CD4 image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg046
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.23 Å Release Date: 2018-08-29
Classification: TRANSCRIPTION/INHIBITOR
Ligands: EX1, EDO

6CIS image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg047
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.51 Å Release Date: 2018-08-29
Classification: TRANSCRIPTION/INHIBITOR
Ligands: X26, EDO, NO3

6CIY image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg069
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.68 Å Release Date: 2018-08-29
Classification: TRANSCRIPTION/INHIBITOR
Ligands: F3J, EDO, NO3

6CJ1 image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg071
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.53 Å Release Date: 2018-08-29
Classification: TRANSCRIPTION/INHIBITOR
Ligands: F2S, FND, EDO, NO3

5WA5 image
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Xmd11-50
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.17 Å Release Date: 2018-07-04
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 4K4, EDO
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