Search Count: 16
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3735967A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, I67, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, I67, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3543105A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, ZN, EDO, GOL, IO5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: SAH, ZN, EDO, GOL, IO5
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830334A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, ZN, GOL, 96I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: EDO, ZN, GOL, 96I
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3852279B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, EDO, GOL, C79 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, EDO, GOL, C79
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Cofactor Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, SAM, GOL, EDO
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAH, LUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAH, LUP
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, EDO, SAM, L0J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, EDO, SAM, L0J
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, SAM, O41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, SAM, O41
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAM, O6A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAM, O6A
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Type 1 Prmt In Complex With The Inhibitor Gsk3368715
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2019-07-10 Classification: ANTITUMOR PROTEIN Ligands: SAH, KZS, GOL, DTT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-10
Ligands: SAH, KZS, GOL, DTT
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SFG, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAM, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, 3XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 3XV
