Search Count: 38,267
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Crystal Structure Of The Yeast 20S Proteasome:Tmc-95A Complex: A Non-Covalent Proteasome Inhibitor
Organism: Saccharomyces cerevisiae, Apiospora montagnei
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2002-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG |
Organism: Saccharomyces cerevisiae, Apiospora montagnei
Method: X-RAY DIFFRACTION
Release Date: 2002-02-13
Ligands: MG
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Crystal Structure Of 20S Proteasome With Novel Inhibitor K-7174
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2013-05-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: WPI |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2013-05-01
Ligands: WPI
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Yeast 20S Proteasome In Complex With Epoxyketone Inhibitor 18
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, MES, 6NV |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, MES, 6NV
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Yeast 20S Proteasome In Complex With Epoxyketone Inhibitor 16
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 79P, MES |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, 79P, MES
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Yeast 20S Proteasome In Complex With Epoxyketone Inhibitor 14
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 6N5, MES |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, 6N5, MES
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Yeast 20S Proteasome In Complex With The Peptidic Epoxyketone Inhibitor 27
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2016-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 6KF, MES |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: MG, CL, 6KF, MES
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Yeast 20S Proteasome In Complex With The Peptidic Epoxyketone Inhibitor 15
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 6KG, MES |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: MG, CL, 6KG, MES
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Ycp In Complex With Tripeptidic Epoxyketone Inhibitor 8
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, MES, 38N |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: MG, MES, 38N
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Ycp In Complex With Tripeptidic Epoxyketone Inhibitor 9
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, MES, 38X |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: MG, MES, 38X
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Ycp In Complex With Tripeptidic Epoxyketone Inhibitor 17
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, MES, 39Q |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: MG, MES, 39Q
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Ycp In Complex With Tripeptidic Epoxyketone Inhibitor 11
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, MES, 37Y |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: MG, MES, 37Y
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Ycp In Complex With Tripeptidic Epoxyketone Inhibitor 2 (Pr924)
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, MES, 39V |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: MG, MES, 39V
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Yeast 20S Proteasome With Human Beta5C (1-138) And Human Beta6 (99-132) In Complex With Epoxyketone Inhibitor 14
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, MES, 6N5 |
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, MES, 6N5
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Yeast 20S Proteasome With Human Beta5C (1-138) And Human Beta6 (97-111; 118-133) In Complex With Epoxyketone Inhibitor 16
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, MES, 79P |
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, MES, 79P
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Yeast 20S Proteasome With Mouse Beta5I (1-138) And Mouse Beta6 (97-111; 118-133) In Complex With Epoxyketone Inhibitor 14
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 6N5, MES |
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, 6N5, MES
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Yeast 20S Proteasome With Human Beta5C (1-138) And Human Beta6 (97-111; 118-133) In Complex With Epoxyketone Inhibitor 17
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 04C, MES |
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, 04C, MES
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Yeast 20S Proteasome With Mouse Beta5I (1-138) And Mouse Beta6 (97-111; 118-133) In Complex With Epoxyketone Inhibitor 18
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 6NV, MES |
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, 6NV, MES
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Yeast 20S Proteasome With Human Beta5C (1-138) And Human Beta6 (97-111; 118-133) In Complex With Epoxyketone Inhibitor 18
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, MES, 6NV |
Organism: Homo sapiens, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, MES, 6NV
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Yeast 20S Proteasome With Mouse Beta5I (1-138) And Mouse Beta6 (97-111; 118-133) In Complex With Epoxyketone Inhibitor 16
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 79P, MES |
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, 79P, MES
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Yeast 20S Proteasome With Mouse Beta5I (1-138) And Mouse Beta6 (97-111; 118-133) In Complex With Epoxyketone Inhibitor 17
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, CL, 79L, MES |
Organism: Mus musculus, Saccharomyces cerevisiae (strain atcc 204508 / s288c), Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: MG, CL, 79L, MES
