Search Count: 20
![]() |
Sars-Cov-2 Main Protease With Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-10-22 Classification: VIRAL PROTEIN, HYDROLASE Ligands: A1B3B, BTB, EDO |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2025-10-22
Ligands: A1B3B, BTB, EDO
![]() |
Sars-Cov-2 Main Protease With Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2025-09-10 Classification: VIRAL PROTEIN Ligands: A1A3N |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1A3N
![]() |
Sars-Cov-2 Main Protease With Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2025-09-10 Classification: VIRAL PROTEIN Ligands: A1A3O |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1A3O
![]() |
Molecular Mechanism Of The The Wake-Promoting Agent Tak-925
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2022-06-08 Classification: SIGNALING PROTEIN Ligands: A6F, OLA |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2022-06-08
Ligands: A6F, OLA
![]() |
Structure Of The Orexin-2 Receptor(Ox2R) Bound To Tak-925, Gi And Scfv16
Organism: Homo sapiens, Bos taurus, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2022-05-25 Classification: MEMBRANE PROTEIN Ligands: OLA, A6F |
Organism: Homo sapiens, Bos taurus, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2022-05-25
Ligands: OLA, A6F
![]() |
Halk In Complex With ((1S,2S)-1-(2,4-Difluorophenyl)-2-(2-(3-Methyl-1H-Pyrazol-5-Yl)-4-(Trifluoromethyl)Phenoxy)Cyclopropyl)Methanamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-01-20 Classification: TRANSFERASE Ligands: W47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: W47
![]() |
Halk In Complex With 1-[(1R,2R)-1-(2,4-Difluorophenyl)-2-[2-(5-Methyl-1H-Pyrazol-3-Yl)-4-(Trifluoromethyl)Phenoxy]Cyclopropyl]Methanamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2021-01-20 Classification: TRANSFERASE Ligands: VTA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: VTA, EDO
![]() |
Halk In Complex With 3-(3-Chlorophenyl)-5-Methyl-1H-Pyrazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2021-01-20 Classification: TRANSFERASE Ligands: VTD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: VTD, EDO
![]() |
Halk In Complex With 3-(3-Methyl-1H-Pyrazol-5-Yl)Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-01-20 Classification: TRANSFERASE Ligands: GOL, VRM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: GOL, VRM
![]() |
Crystal Structure Of Tyk2 With Novel Pyrrolidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2020-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: N9G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: N9G
![]() |
Structure Of Tyk2 With Inhibitor 16: 3-Azanyl-5-[(2~{S})-3-Methylbutan-2-Yl]-7-[1-Methyl-5-(2-Oxidanylpropan-2-Yl)Pyrazol-3-Yl]-1~{H}-Pyrazolo[4,3-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2016-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5U3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-13
Ligands: 5U3
![]() |
Structure Of Tyk2 With Inhibitor 4: 3-Azanyl-5-(2-Methylphenyl)-7-(1-Methylpyrazol-3-Yl)-1~{H}-Pyrazolo[4,3-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2016-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5U4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-13
Ligands: 5U4
![]() |
X-Ray Structure Of Endolysin From Clostridium Perfringens Phage Phism101
Organism: Clostridium phage phism101
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2014-04-02 Classification: HYDROLASE Ligands: EPE, ACT, MLA |
Organism: Clostridium phage phism101
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: EPE, ACT, MLA
![]() |
X-Ray Structure Of Catalytic Domain Of Endolysin From Clostridium Perfringens Phage Phism101
Organism: Clostridium phage phism101
Method: X-RAY DIFFRACTION Resolution:1.37 Å Release Date: 2014-04-02 Classification: HYDROLASE Ligands: NDG, NAG, PO4 |
Organism: Clostridium phage phism101
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: NDG, NAG, PO4
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Hinge Binding Pyrazolobenzothiazine Compound.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-03-06 Classification: transferase/transferase inhibitor Ligands: 1BQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: 1BQ
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With An Allosteric Binding Pyrazolobenzothiazine Compound.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-02-06 Classification: transferase/transferase inhibitor Ligands: IPA, 1BR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-06
Ligands: IPA, 1BR
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Novel Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2012-08-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0O7, IPA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-22
Ligands: 0O7, IPA
![]() |
Structure Of Focal Adhesion Kinase Catalytic Domain In Complex With Novel Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-07-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0PF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-25
Ligands: 0PF
![]() |
Crystal Structure Of Clostridium Histolyticum Colg Collagenase Collagen-Binding Domain 3B At 1.65 Angstrom Resolution In Presence Of Calcium
Organism: Clostridium histolyticum
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2003-04-15 Classification: HYDROLASE Ligands: CA |
Organism: Clostridium histolyticum
Method: X-RAY DIFFRACTION
Release Date: 2003-04-15
Ligands: CA
![]() |
Crystal Structure Of Clostridium Histolyticum Colg Collagenase Collagen-Binding Domain 3B At 1.0 Angstrom Resolution In Absence Of Calcium
Organism: Clostridium histolyticum
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2003-04-15 Classification: HYDROLASE Ligands: CL, LI |
Organism: Clostridium histolyticum
Method: X-RAY DIFFRACTION
Release Date: 2003-04-15
Ligands: CL, LI
