Search Count: 18
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Bacterial Cereblon Homologue In Complex With (R)-3-(4-Methoxyphenyl)Piperidine-2,6-Dione
Organism: Magnetospirillum gryphiswaldense
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-04-13 Classification: SIGNALING PROTEIN Ligands: ZN, 9FT |
Organism: Magnetospirillum gryphiswaldense
Method: X-RAY DIFFRACTION
Release Date: 2022-04-13
Ligands: ZN, 9FT
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Crystal Structure Of The Second Bromodomain Of Human Brd2 In Complex With The Compound 3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2021-11-17 Classification: TRANSCRIPTION Ligands: EDO, YA3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: EDO, YA3
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Braf In Complex With N-(4-Methyl-3-(1-Methyl-2-Oxo-2,3-Dihydro-1H-Benzo[D]Imidazol-5-Yl)Phenyl)-3-(Trifluoromethyl)Benzamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2019-10-23 Classification: transferase/transferase inhibitor Ligands: K7S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: K7S
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Braf In Complex With N-(3-(2-(2-Hydroxyethoxy)-6-Morpholinopyridin-4-Yl)-4-Methylphenyl)-2-(Trifluoromethyl)Isonicotinamide (Lxh254)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2019-09-04 Classification: transferase/transferase inhibitor Ligands: K81 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K81
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp244
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2018-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DZV, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: DZV, PO4, GOL
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitors Shp099 And Shp244
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2018-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 5OD, DZV, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: 5OD, DZV, PO4, GOL
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp504
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DZS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: DZS, PO4
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitors Shp099 And Shp504
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 5OD, DZS, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: 5OD, DZS, PO4, GOL
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2018-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DYV, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: DYV, PO4, GOL
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitors Shp099 And Shp844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2018-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 5OD, DYV, PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: 5OD, DYV, PO4, GOL
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Braf In Complex With N-(3-(Tert-Butyl)Phenyl)-4-Methyl-3-(6-Morpholinopyrimidin-4-Yl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 92D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 92D
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Braf In Complex With Raf709
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 92J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 92J
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Design, Synthesis And Structure Activity Relationship Of Potent Pan-Pim Kinase Inhibitors Derived From The Pyridyl-Amide Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-04-06 Classification: Transferase/Transferase Inhibitor Ligands: PEG, 6CB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: PEG, 6CB
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Identification Of N-(4-((1R,3S,5S)-3-Amino-5-Methylcyclohexyl)Pyridin-3-Yl)-6-(2,6-Difluorophenyl)-5-Fluoropicolinamide (Pim447), A Potent And Selective Proviral Insertion Site Of Moloney Murine Leukemia (Pim) 1,2 And 3 Kinase Inhibitor In Clinical Trials For Hematological Malignancies
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-11-11 Classification: Transferase/Transferase Inhibitor Ligands: 5H7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 5H7
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Pim1 Complexed With A Phenylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HV
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Pim1 Complexed With A Pyridylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HW, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HW, GOL
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Pim1 Complexed With A Pyridylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HX
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Pim1 Complexed With A Novel 3,6-Disubstituted Indole At 2.6 Ang Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-10-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3T9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: 3T9