Search Count: 14
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Crystal Structure Of Human Glutaminyl Cyclase In Complex With N-(2-(1H-Imidazol-5-Yl)Ethyl)-4-Methoxybenzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: ZN, A1EFY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: ZN, A1EFY
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Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With The Inhibitor N-(1H-Benzo[D]Imidazol-5-Yl)-1-Phenylmethanesulfonamide (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2025-03-12 Classification: TRANSFERASE Ligands: ZN, A1D93, GOL, DMS, DMF, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-12
Ligands: ZN, A1D93, GOL, DMS, DMF, PEG
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Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With The Inhibitor 3-((2-(1H-Imidazol-5-Yl)Ethyl)Carbamoyl)-4-Amino-1,2,5-Oxadiazole 2-Oxide (Compound 13)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2025-03-12 Classification: TRANSFERASE Ligands: ZN, A1D94, DMS, GOL, DMF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-12
Ligands: ZN, A1D94, DMS, GOL, DMF
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Crystal Structure Of Human Golgi Resident Glutaminyl Cyclase In Complex With (Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-(Piperidin-4-Yloxy)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.13 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D46 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: ZN, A1D46
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Crystal Structure Of Human Golgi Resident Glutaminyl Cyclase In Complex With (Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-((Tetrahydro-2H-Pyran-4-Yl)Oxy)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.54 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: ZN, A1D47
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Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With (S)-1-(1H-Benzo[D]Imidazol-5-Yl)-5-(4-Propoxyphenyl)Imidazolidin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.24 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: ZN, A1D49
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Crystal Structure Of Human Secretory Glutaminyl Cyclase In Complex With (Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-Hydroxyindolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D48 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: ZN, A1D48
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Crystal Structure Of Human Golgi Resident Glutaminyl Cyclase In Complex With (R,Z)-3-((1H-Benzo[D]Imidazol-5-Yl)Methylene)-4-((1-Acetylpyrrolidin-3-Yl)Oxy)Indolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2024-06-12 Classification: TRANSFERASE Ligands: ZN, A1D5C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-12
Ligands: ZN, A1D5C
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Crystal Structure Of Human Indoleamine 2,3-Dioxygenagse 1 (Hido1) Complexed With 6-Bromo-1H-Indazol-4-Amine (1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2021-07-21 Classification: OXIDOREDUCTASE Ligands: HS0, HEM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: HS0, HEM
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Crystal Structure Of Human Indoleamine 2,3-Dioxygenagse 1 (Hido1) Complexed With 4-(((6-Bromo-1H-Indazol-4-Yl)Amino)Methyl)Phenol (2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2021-07-21 Classification: OXIDOREDUCTASE Ligands: HU0, HEM, ACY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: HU0, HEM, ACY
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Crystal Structure Of Human Indoleamine 2,3-Dioxygenagse 1 (Hido1) Complexed With (1S,2R)-2-(((6-Bromo-1H-Indazol-4-Yl)Amino)Methyl)Cyclohexan-1-Ol (22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2021-07-21 Classification: OXIDOREDUCTASE Ligands: HEM, HU3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: HEM, HU3
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Crystal Structure Of Human Indoleamine 2,3-Dioxygenagse 1 (Hido1) Complexed With (1R,2S)-2-(((6-Bromo-1H-Indazol-4-Yl)Amino)Methyl)Cyclohexan-1-Ol (23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2021-07-21 Classification: OXIDOREDUCTASE Ligands: HEM, HU6, ACY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: HEM, HU6, ACY
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Crystal Structure Of Human Indoleamine 2,3-Dioxygenagse 1 (Hido1) Complexed With (1R,2S)-2-(((5-Bromo-1H-Indazol-4-Yl)Amino)Methyl)Cyclohexan-1-Ol (36)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2021-07-21 Classification: OXIDOREDUCTASE Ligands: HEM, HU9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: HEM, HU9
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Crystal Structure Of Human Indoleamine 2,3-Dioxygenagse 1 (Hido1) Complexed With 6-Bromo-N-(((1S,2S)-2-Chlorocyclohexyl)Methyl)-1H-Indazol-4-Amine (39)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-07-21 Classification: OXIDOREDUCTASE Ligands: HEM, HUC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-21
Ligands: HEM, HUC