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8CDW image
Crystal Structure Of Human Hpk1 (Map4K1) Complex With 7-(1-Methyl-1H-Pyrazol-4-Yl)-N-[4-(1-Methylpiperidin-4-Yl)Phenyl]Quinazolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2023-08-16
Classification: TRANSFERASE
Ligands: UES

8CIJ image
Crystal Structure Of Human Hpk1 (Map4K1) Complex With 2-[8-Amino-7-Fluoro-6-(8-Methyl-2,3-Dihydro-1H-Pyrido[2,3-B][1,4]Oxazin-7-Yl)-Isoquinolin-3-Ylamino]-6-Isopropyl-5,6-Dihydro-4H-1,6,8A-Triaza-Azulen-7-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.82 Å Release Date: 2023-08-16
Classification: TRANSFERASE
Ligands: USF

7N91 image
P70 S6K1 In Complex With Msc2317067A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.00 Å Release Date: 2022-07-06
Classification: TRANSFERASE/INHIBITOR
Ligands: 1RJ

7N93 image
P70 S6K1 In Complex With Msc2363318A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.74 Å Release Date: 2022-07-06
Classification: TRANSFERASE/INHIBITOR
Ligands: 1SK

7KXL image
Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.84 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9J, DMS

7KXM image
Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.33 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9M

7KXN image
Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.34 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9P, DMS

7KXO image
Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.94 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9S, DMS

7KXP image
Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.83 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: X9V, DMS

7KXQ image
Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.38 Å Release Date: 2021-05-19
Classification: TRANSFERASE
Ligands: DMS, X9Y

6DI0 image
Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.30 Å Release Date: 2018-10-17
Classification: TRANSFERASE/TRANSFERASE Inhibitor
Ligands: GJG

6DI1 image
Crystal Structure Of Btk In Complex With Covalent Fragment Ligand
Organism: homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.10 Å Release Date: 2018-10-17
Classification: TRANSFERASE/TRANSFERASE inhibitor
Ligands: GJD

6DI3 image
Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2018-09-05
Classification: TRANSFERASE/TRANSFERASE Inhibitor
Ligands: GJA

6DI5 image
Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.42 Å Release Date: 2018-09-05
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: GJ7, DMS

6DI9 image
Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.25 Å Release Date: 2018-09-05
Classification: TRANSFERASE/TRANSFERASE Inhibitor
Ligands: GJJ, DMS
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