Search Count: 15
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Crystal Structure Of Human Hpk1 (Map4K1) Complex With 7-(1-Methyl-1H-Pyrazol-4-Yl)-N-[4-(1-Methylpiperidin-4-Yl)Phenyl]Quinazolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2023-08-16 Classification: TRANSFERASE Ligands: UES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-16
Ligands: UES
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Crystal Structure Of Human Hpk1 (Map4K1) Complex With 2-[8-Amino-7-Fluoro-6-(8-Methyl-2,3-Dihydro-1H-Pyrido[2,3-B][1,4]Oxazin-7-Yl)-Isoquinolin-3-Ylamino]-6-Isopropyl-5,6-Dihydro-4H-1,6,8A-Triaza-Azulen-7-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2023-08-16 Classification: TRANSFERASE Ligands: USF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-16
Ligands: USF
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P70 S6K1 In Complex With Msc2317067A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2022-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: 1RJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: 1RJ
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P70 S6K1 In Complex With Msc2363318A-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2022-07-06 Classification: TRANSFERASE/INHIBITOR Ligands: 1SK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: 1SK
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9J, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9J, DMS
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9M
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Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9P, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9P, DMS
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Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9S, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9S, DMS
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Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9V, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9V, DMS
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Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: DMS, X9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: DMS, X9Y
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Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-17 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: GJG
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Crystal Structure Of Btk In Complex With Covalent Fragment Ligand
Organism: homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2018-10-17 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: GJD |
Organism: homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: GJD
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Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJA
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Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GJ7, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJ7, DMS
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Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJJ, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJJ, DMS
