Search Count: 20
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Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, NAG, A1JCF, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, NAG, A1JCF, PO4
 |
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, NAG, A1JCG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, NAG, A1JCG, PO4
 |
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 6 (Oric-533)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, A1JCH, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, A1JCH, PO4
 |
Crystal Structure Of Pak1 In Complex With An Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-09-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 59N
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Crystal Structure Of P21-Activated Kinase 1 (Pak1) In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2016-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: 6BZ
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound G-5555
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59T
 |
Crystal Structure Of Pak1 In Complex With An Inhibitor Compound Frax1036
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59U, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59U, DMS
 |
Apo Mitogen-Activated Protein Kinase Kinase Kinase Kinase 4 (Map4K4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-01-06 Classification: TRANSFERASE Ligands: DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-06
Ligands: DMS
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Apo Map4K4 T181E Phosphomimetic Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2016-01-06 Classification: TRANSFERASE Ligands: MES, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-06
Ligands: MES, NA
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Mitogen-Activated Protein Kinase Kinase Kinase Kinase 4 (Map4K4) Bound To Amppnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-01-06 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-06
Ligands: ANP, MG
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Map4K4 Bound To Inhibitor Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-06 Classification: Transferase/Transferase inhibitor Ligands: 3C8, MG, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-06
Ligands: 3C8, MG, MES
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Map4K4 T181E Mutant Bound To Inhibitor Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-01-06 Classification: Transferase/Transferase inhibitor Ligands: MES, 3C8, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-06
Ligands: MES, 3C8, MG
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Map4K4 In Complex With Inhibitor Gne-495
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2015-09-02 Classification: Transferase/Transferase Inhibitor Ligands: MG, MES, 4P4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: MG, MES, 4P4
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Discovery Of A Potent And Selective Bcl-Xl Inhibitor That Demonstrates Thrombocytopenia And Inhibits Tumor Growth In Vivo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-07-22 Classification: APOPTOSIS/INHIBITOR Ligands: 3CQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: 3CQ
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Map4K4 In Complex With Inhibitor (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: 3D8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 3D8
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Map4K4 In Complex With Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: MES, NA, 3D9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: MES, NA, 3D9
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Map4K4 In Complex With Inhibitor (Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-09-03 Classification: Transferase/Transferase inhibitor Ligands: MG, 3DC, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: MG, 3DC, MES
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Map4K4 In Complex With Inhibitor (Compound 22), 6-(3-Chlorophenyl)Quinazolin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MES, NA, 2QV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MES, NA, 2QV
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Map4K4 In Complex With Inhibitor (Compound 29), 6-(2-Fluoropyridin-4-Yl)Pyrido[3,2-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MG, MES, 2QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MG, MES, 2QU
 |
Map4K4 In Complex With Inhibitor (Compound 31), N-[3-(4-Aminoquinazolin-6-Yl)-5-Fluorophenyl]-2-(Pyrrolidin-1-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2014-04-23 Classification: transferase/transferase inhibitor Ligands: MES, MG, 2QT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-23
Ligands: MES, MG, 2QT