Search Count: 18
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Crystal Structure Of Pi3K-Alpha In Complex With Taselisib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: 799 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: 799
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3W
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3R
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Crystal Structure Of Pi3K-Alpha In Complex With Compound 32
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-11-30 Classification: CELL CYCLE Ligands: X3N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-30
Ligands: X3N
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Chk1 Kinase Domain With Diazacarbazole Compound 8: N-[3-(6-Cyano-9H-Pyrrolo[2,3-B:5,4-C']Dipyridin-3-Yl)Phenyl]Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3XK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3XK
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Chk1 Kinase Domain With Diazacarbazole Compound 7: 3-(2-Hydroxyphenyl)-9H-Pyrrolo[2,3-B:5,4-C']Dipyridine-6-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3XL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3XL
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Chk1 Kinase Domain With Diazacarbazole Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-06-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3X7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 3X7
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The Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-05-22 Classification: TRANSFERASE Ligands: C5I, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: C5I, EDO
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Jak2 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-[(8As)-2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(8Ah)-Yl]Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor (Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexyl)Acetonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J6
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 15T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 15T
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NH
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Jak2 Kinase (Jh1 Domain) In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NH
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NL
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NT, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NT, PEG
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Jak2 Kinase (Jh1 Domain) Triple Mutant In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NU, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NU, GOL
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Jak2 Kinase (Jh1 Domain) Triple Mutant In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0NV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0NV