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3ZBX image
X-Ray Structure Of C-Met Kinase In Complex With Inhibitor 6-((6-(4- Fluorophenyl)-(1,2,4)Triazolo(4,3-B)(1,2,4)Triazin-3-Yl)Methyl) Quinoline.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2013-11-27
Classification: TRANSFERASE
Ligands: 6XE

3ZC5 image
X-Ray Structure Of C-Met Kinase In Complex With Inhibitor (S)-6-(1-(6- (1-Methyl-1H-Pyrazol-4-Yl)-(1,2,4)Triazolo(4,3-B)Pyridazin-3-Yl)Ethyl) Quinoline.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2013-11-27
Classification: TRANSFERASE
Ligands: W9Z

3ZCL image
X-Ray Structure Of C-Met Kinase In Complex With Inhibitor (S)-3-(1-(1H-Pyrrolo(2,3-B)Pyridin-3-Yl)Ethyl)-N-Isopropyl-(1,2,4)Triazolo(4,3- B)Pyridazin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.40 Å Release Date: 2013-11-27
Classification: TRANSFERASE
Ligands: 5TF

4AOI image
Crystal Structure Of C-Met Kinase Domain In Complex With 4-(3-((1H- Pyrrolo(2,3-B)Pyridin-3-Yl)Methyl)-(1,2,4)Triazolo(4,3-B)(1,2,4) Triazin-6-Yl)Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2012-09-26
Classification: TRANSFERASE
Ligands: 4K0

4AP7 image
Crystal Structure Of C-Met Kinase Domain In Complex With 4-((6-(4- Fluorophenyl)-(1,2,4)Triazolo(4,3-B)(1,2,4)Triazin-3-Yl)Methyl)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2012-09-26
Classification: TRANSFERASE
Ligands: F47

3ZZE image
Crystal Structure Of C-Met Kinase Domain In Complex With N'-((3Z)-4- Chloro-7-Methyl-2-Oxo-1,2-Dihydro-3H-Indol-3-Ylidene)-2-(4- Hydroxyphenyl)Propanohydrazide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.87 Å Release Date: 2011-09-14
Classification: TRANSFERASE
Ligands: 6XP

3ZXZ image
X-Ray Structure Of Pf-04217903 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2011-08-31
Classification: TRANSFERASE
Ligands: KRW

3OAW image
4-Methylpteridineones As Orally Active And Selective Pi3K/Mtor Dual Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.75 Å Release Date: 2010-09-22
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: OAW

2XP2 image
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With Crizotinib (Pf-02341066)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2010-09-15
Classification: TRANSFERASE
Ligands: VGH

2WKM image
X-Ray Structure Of Pha-00665752 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2010-08-25
Classification: TRANSFERASE
Ligands: PFY

2WGJ image
X-Ray Structure Of Pf-02341066 Bound To The Kinase Domain Of C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2009-06-02
Classification: TRANSFERASE
Ligands: VGH
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