Search Count: 6
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Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2017-11-29 Classification: Transferase/Transferase Inhibitor Ligands: YAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-29
Ligands: YAM
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Selectivity Switch Between Fak And Pyk2: Macrocyclization Of Fak Inhibitors Improves Pyk2 Potency
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-12-21 Classification: Transferase/Transferase Inhibitor Ligands: 7FM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: 7FM
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Crystal Structure Of An Optimzied Benzothiophene Inhibitor Bound To Mapkap Kinase-2 (Mk-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.80 Å Release Date: 2009-04-07 Classification: TRANSFERASE Ligands: B97 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: B97
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Crystal Structure Of A Benzthiophene Lead Bound To Mapkap Kinase-2 (Mk-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2009-04-07 Classification: TRANSFERASE Ligands: B98 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: B98
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Crystal Structure Of A Benzthiophene Inhibitor Bound To Human Cyclin-Dependent Kinase-2 (Cdk-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-04-07 Classification: TRANSFERASE Ligands: B98 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: B98
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Crystal Structure Of A Pyrrolopyridine Inhibitor Bound To Mapkap Kinase-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.80 Å Release Date: 2007-06-12 Classification: TRANSFERASE Ligands: F10 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-06-12
Ligands: F10
