Search Count: 6
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From Dna-Encoded Library Screening To Am-9747 - An Mta-Cooperative Prmt5 Inhibitor With Potent Oral In Vivo Efficacy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2025-03-26 Classification: TRANSFERASE/INHIBITOR Ligands: A1BQW, MTA, GOL, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-26
Ligands: A1BQW, MTA, GOL, PEG, DMS
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Amg 193, A Clinical Stage Mta-Cooperative Prmt5 Inhibitor, Drives Anti-Tumor Activity Preclinically And In Patients With Mtap-Deleted Cancers
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2024-10-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, DMS, A1ATH, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GOL, DMS, A1ATH, MTA
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X-Ray Structure Of C-Met With Triazolopyridazine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2008-04-29 Classification: TRANSFERASE Ligands: LKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-29
Ligands: LKG
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X-Ray Structure Of C-Met With Triazolopyridazine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-04-29 Classification: TRANSFERASE Ligands: L5G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-29
Ligands: L5G
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X-Ray Structure Of C-Met With Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-11-06 Classification: TRANSFERASE Ligands: AM7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: AM7
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X-Ray Structure Of Su11274 Bound To C-Met
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-11-06 Classification: TRANSFERASE Ligands: AM8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: AM8
