Search Count: 5
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Crystal Structure Of The Mertk Kinase Domain With Sa4488
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2024-10-09 Classification: TRANSFERASE Ligands: A1APF, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APF, CL
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Mertk In Complex With Small Molecule 6-{1-[([1,1'-Biphenyl]-4-Yl)Carbamoyl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APG, CL
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Mertk In Complex With Small Molecule Inhibitor 6-{1-[6-(3-Hydroxy-3-Methylbutoxy)-1,3-Benzoxazol-2-Yl]Azetidin-3-Yl}-3-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]Pyrazine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-10-09 Classification: TRANSFERASE/INHIBITOR Ligands: A1APH, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-09
Ligands: A1APH, CL
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The Novel P300/Cbp Inhibitor A-485 Uncovers A Unique Mechanism Of Action To Target Ar In Castrate Resistant Prostate Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-09-27 Classification: transferase/transferase INHIBITOR Ligands: 6TF, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: 6TF, NA
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Nmr Structure Of The Substrate Binding Domain Of Dnak In The Apo Form
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Organism: Escherichia coli
Method: SOLUTION NMR
Release Date: 1999-12-08
