Search Count: 16
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Identification Of Low Micromolar Sars-Cov-2 Mpro Inhibitors From Hits Identified By In Silico Screens
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-05-04 Classification: HYDROLASE Ligands: 4N0 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: 4N0
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Discovery Of 5,6,7,8-Tetrahydropyrido[3,4-D]Pyrimidine Inhibitors Of Erk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-05-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2SH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-21
Ligands: 2SH
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Human Trka In Complex With The Inhibitor Az-23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2012-08-15 Classification: TRANSFERASE Ligands: V4Z, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: V4Z, ZN
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Orally Active Aminopyridines As Inhibitors Of Tetrameric Fructose 1,6- Bisphosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: YCU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: YCU
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Orally Active Aminopyridines As Inhibitors Of Tetrameric Fructose 1,6- Bisphosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: RO8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: RO8
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Fructose-1,6-Bisphosphatase(D-Fructose-1,6-Bisphosphate-1- Phosphohydrolase) (E.C.3.1.3.11) Complexed With An Amp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: RO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: RO3
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Fructose-1,6-Bisphosphatase(D-Fructose-1,6-Bisphosphate-1- Phosphohydrolase) (E.C.3.1.3.11) Complexed With An Amp Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-12-22 Classification: HYDROLASE Ligands: RO5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-12-22
Ligands: RO5
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Design And Biological Evaluation Of Novel, Balanced Dual Ppara/G Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-10-20 Classification: TRANSCRIPTION Ligands: CTM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-20
Ligands: CTM
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Design And Biological Evaluation Of Novel, Balanced Dual Ppara/G Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2009-10-20 Classification: TRANSCRIPTION Ligands: CTM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-20
Ligands: CTM
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Hepatitis C Virus Polymerase Ns5B (Bk 1-570) With Thiazine Inhibitor
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-09-08 Classification: TRANSFERASE Ligands: T18, NI |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2009-09-08
Ligands: T18, NI
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Hepatitis C Virus Polymerase Ns5B With Thiazine Inhibitor 2
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-09-08 Classification: TRANSFERASE Ligands: H59 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2009-09-08
Ligands: H59
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Hepatitis C Virus Polymerase Ns5B With Saccharin Inhibitor
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-09-08 Classification: TRANSFERASE Ligands: H5S |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2009-09-08
Ligands: H5S
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Hepatitis C Virus Polymerase Ns5B With Saccharin Inhibitor 1
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-09-08 Classification: TRANSFERASE Ligands: H5U |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2009-09-08
Ligands: H5U
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Aleglitazar, A New, Potent, And Balanced Ppar Alpha/Gamma Agonist For The Treatment Of Type Ii Diabetes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-06-02 Classification: TRANSCRIPTION/TRANSFERASE Ligands: RO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-02
Ligands: RO7
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Aleglitaar. A New. Potent, And Balanced Dual Ppara/G Agonist For The Treatment Of Type Ii Diabetes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-06-02 Classification: TRANSCRIPTION/TRANSFERASE Ligands: RO7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-02
Ligands: RO7
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Structure-Based Design Of Indole Propionic Acids As Novel Pparag Co-Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-09-26 Classification: TRANSCRIPTION REGULATOR Ligands: 208 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-26
Ligands: 208