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Search Count: 8

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6ALJ image
Aldh1A2 Liganded With Nad And Compound Win18,446
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.89 Å Release Date: 2018-01-10
Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR
Ligands: NAD, CW2

6B5G image
Aldh1A2 Liganded With Nad And (3-Ethoxythiophen-2-Yl){4-[4-Nitro-3-(Pyrrolidin-1-Yl)Phenyl]Piperazin-1-Yl}Methanone (Compound 6-118)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2018-01-10
Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR
Ligands: NAD, CQY

6B5H image
Aldh1A2 Liganded With Nad And 1-(4-Cyanophenyl)-N-(3-Fluorophenyl)-3-[4-(Methylsulfonyl)Phenyl]-1H-Pyrazole-4-Carboxamide (Compound Cm121)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2018-01-10
Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR
Ligands: NAD, CU4

6B5I image
Aldh1A2 Liganded With 1-(4-Cyanophenyl)-N-(3-Fluorophenyl)-3-[4-(Methylsulfonyl)Phenyl]-1H-Pyrazole-4-Carboxamide (Compound Cm121)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2018-01-10
Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR
Ligands: CU4

5MT6 image
Structure Of E.Coli Glpg In Complex With Peptide Derived Inhibitor Ac-Rvrha-Phenylethyl-Ketoamide
Organism: Escherichia coli k-12, Providencia stuartii
Method: X-RAY DIFFRACTION
Resolution:2.16 Å Release Date: 2017-11-15
Classification: HYDROLASE
Ligands: BNG

5MT7 image
Structure Of E.Coli Glpg In Complex With Peptide Derived Inhibitor Ac-Vrha-Cmk
Organism: Escherichia coli k-12, Providencia stuartii
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2017-11-15
Classification: HYDROLASE

5MT8 image
Structure Of E.Coli Glpg In Complex With Peptide Derived Inhibitor Ac-Rvrha-Cmk
Organism: Escherichia coli k-12, Providencia stuartii
Method: X-RAY DIFFRACTION
Resolution:1.95 Å Release Date: 2017-11-15
Classification: HYDROLASE
Ligands: BNG, CL

5MTF image
A Modular Route To Novel Potent And Selective Inhibitors Of Rhomboid Intramembrane Proteases
Organism: Escherichia coli o45:k1 (strain s88 / expec), Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:1.79 Å Release Date: 2017-11-15
Classification: HYDROLASE
Ligands: CL, BNG
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