Search Count: 29
![]() |
Wild-Type Menin Complexed With Jnj-75276617
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 9N6, EDO, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 9N6, EDO, MG, NA
![]() |
[M322I] Menin Complexed With Jnj-75276617
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 9N6, EDO, MG, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 9N6, EDO, MG, MES
![]() |
Wild-Type Menin Complexed With Ds-1594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 7IX, EDO, NA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 7IX, EDO, NA, MG
![]() |
[M322I] Menin Complexed With Ds-1594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 7IX, EDO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 7IX, EDO, MG
![]() |
Wild-Type Menin Complexed With Dsp-5336
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 2IZ, EDO, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 2IZ, EDO, MG, GOL
![]() |
[M322I] Menin Complexed With Dsp-5336
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 2IZ, EDO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 2IZ, EDO, MG
![]() |
Wild-Type Menin Complexed With Ko-539
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: K5O, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: K5O, MG
![]() |
[M322I] Menin Complexed With Ko-539
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: EDO, K5O, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: EDO, K5O, MG
![]() |
Inhibition Of Human Menin By Vtp-50469
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-12-18 Classification: TRANSCRIPTION Ligands: OP4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: OP4
![]() |
Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y4
![]() |
Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y8
![]() |
Discovery Of Novel, Orally Efficacious Liver X Receptor (Lxr) Beta Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2016-06-29 Classification: DNA BINDING PROTEIN Ligands: 67S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 67S
![]() |
Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, CL, RX5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: NAG, CL, RX5
![]() |
Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, RX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: CL, RX6
![]() |
Alkyl Amine Renin Inhibitors: Filling S1 From S3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RX0, GOL, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: RX0, GOL, NAG
![]() |
Optimization Of Orally Bioavailable Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-01-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 22X, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: 22X, NAG
![]() |
Crystal Structure Of Human Flap With Mk-591
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:4.25 Å Release Date: 2007-08-21 Classification: MEMBRANE PROTEIN, LIPID TRANSPORT Ligands: 2CS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-21
Ligands: 2CS
![]() |
Crystal Structure Of Human Flap With An Iodinated Analog Of Mk-591
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:4.00 Å Release Date: 2007-08-21 Classification: MEMBRANE PROTEIN, LIPID TRANSPORT Ligands: 3CS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-21
Ligands: 3CS
![]() |
Human Estrogen Receptor Beta Ligand-Binding Domain In Complex With Compound 45
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2006-10-10 Classification: TRANSCRIPTION REGULATOR Ligands: FBR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-10-10
Ligands: FBR
![]() |
Crystal Structure Of Human Ppar-Gamma Ligand Binding Domain Complexed With An Alpha-Aryloxyphenylacetic Acid Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-04-25 Classification: TRANSCRIPTION Ligands: C01 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-04-25
Ligands: C01
