Search Count: 43
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Structure Of Bovine Endothelial Nitric Oxide Synthase Heme Domain In Complex With 6-Acetyl-2-Amino-7,7-Dimethyl-7,8-Dihydropteridin-4(3H)-One
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2014-05-28 Classification: OXIDOREDUCTASE Ligands: ARG, HEM, WSD, ACT |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: ARG, HEM, WSD, ACT
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Structure Of Bovine Endothelial Nitric Oxide Synthase Heme Domain In Complex With (9As)-2-Amino-9A-Methyl-6,7,8,9,9A,10-Hexahydrobenzo[G]Pteridin-4(3H)-One
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2014-05-28 Classification: OXIDOREDUCTASE Ligands: ARG, HEM, WS7, ACT, ZN, GOL |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: ARG, HEM, WS7, ACT, ZN, GOL
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Structure Of Bovine Endothelial Nitric Oxide Synthase Heme Domain In Complex With (9As)-2-Amino-9A-Methyl-8,9,9A,10-Tetrahydrobenzo[G]Pteridine-4,6(3H,7H)-Dione
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2014-05-28 Classification: OXIDOREDUCTASE Ligands: ARG, HEM, WS6, ACT, GOL, ZN |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: ARG, HEM, WS6, ACT, GOL, ZN
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Structure Of Bovine Endothelial Nitric Oxide Synthase Heme Domain (H4B-Free) Supplemented With 50Um Zn Acetate And With Poor Binding Of 6-Acetyl-2-Amino-7,7-Dimethyl-7,8-Dihydropteridin-4(3H)-One.
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2014-05-28 Classification: OXIDOREDUCTASE Ligands: ARG, HEM, ACT, ZN, GOL |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2014-05-28
Ligands: ARG, HEM, ACT, ZN, GOL
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Discovery And Characterisation Of 2-Anilino-4-(Thiazol-5-Yl) Pyrimidine Transcriptional Cdk Inhibitors As Anticancer Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-11-10 Classification: TRANSFERASE Ligands: CDK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: CDK
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Discovery And Characterisation Of 2-Anilino-4-(Thiazol-5-Yl) Pyrimidine Transcriptional Cdk Inhibitors As Anticancer Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2010-11-10 Classification: TRANSFERASE Ligands: Y8L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: Y8L
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Truncation And Optimisation Of Peptide Inhibitors Of Cdk2, Cyclin A Through Structure Guided Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2010-02-16 Classification: CELL CYCLE Ligands: X1N |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2010-02-16
Ligands: X1N
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Truncation And Optimisation Of Peptide Inhibitors Of Cdk2, Cyclin A Through Structure Guided Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-06-09 Classification: TRANSFERASE Ligands: CK7 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-06-09
Ligands: CK7
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Truncation And Optimisation Of Peptide Inhibitors Of Cdk2, Cyclin A Through Structure Guided Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2009-06-09 Classification: TRANSFERASE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-06-09
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Truncation And Optimisation Of Peptide Inhibitors Of Cdk2, Cyclin A Through Structure Guided Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2009-06-09 Classification: TRANSFERASE |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-06-09
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Replace: A Strategy For Iterative Design Of Cyclin Binding Groove Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-01-29 Classification: TRANSFERASE Ligands: C35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: C35
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Replace: A Strategy For Iterative Design Of Cyclin Binding Groove Inhibitors
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2007-03-27 Classification: TRANSFERASE/INHIBITOR Ligands: MTZ, GVC |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2007-03-27
Ligands: MTZ, GVC
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Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-03-01 Classification: TRANSFERASE Ligands: CK8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-01
Ligands: CK8
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Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-03-01 Classification: TRANSFERASE Ligands: CK2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-01
Ligands: CK2
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Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2006-03-01 Classification: CELL CYCLE Ligands: CK4 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2006-03-01
Ligands: CK4
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Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2006-03-01 Classification: TRANSFERASE/INHIBITOR Ligands: MTW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-01
Ligands: MTW
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Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2006-03-01 Classification: TRANSFERASE Ligands: MTW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-01
Ligands: MTW
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Nmr Structure Of Unliganded Mdm2
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2005-06-28
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Structural And Biochemical Studies Of Human Pcna Complexes Provide The Basis For Association With Cdk/Cyclin And Rationale For Inhibitor Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2005-01-13 Classification: DNA BINDING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-13
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Native Human Pcna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2005-01-13 Classification: DNA BINDING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-01-13
