Search Count: 22
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Wild-Type Menin Complexed With Jnj-75276617
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 9N6, EDO, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 9N6, EDO, MG, NA
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[M322I] Menin Complexed With Jnj-75276617
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 9N6, EDO, MG, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 9N6, EDO, MG, MES
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Wild-Type Menin Complexed With Ds-1594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 7IX, EDO, NA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 7IX, EDO, NA, MG
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[M322I] Menin Complexed With Ds-1594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 7IX, EDO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 7IX, EDO, MG
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Wild-Type Menin Complexed With Dsp-5336
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 2IZ, EDO, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 2IZ, EDO, MG, GOL
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[M322I] Menin Complexed With Dsp-5336
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: 2IZ, EDO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: 2IZ, EDO, MG
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Wild-Type Menin Complexed With Ko-539
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: K5O, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: K5O, MG
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[M322I] Menin Complexed With Ko-539
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-29 Classification: TRANSCRIPTION Ligands: EDO, K5O, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: EDO, K5O, MG
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Inhibition Of Human Menin By Sndx-5613
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-12-14 Classification: TRANSCRIPTION Ligands: OQ4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: OQ4, MG
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Inhibition Of Human Menin By Sndx-5613
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2022-12-14 Classification: TRANSCRIPTION Ligands: OQ4, EDO, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-14
Ligands: OQ4, EDO, MES
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Inhibition Of Human Menin By Vtp-50469
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-12-18 Classification: TRANSCRIPTION Ligands: OP4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: OP4
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y4
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y8
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Discovery Of Novel, Orally Efficacious Liver X Receptor (Lxr) Beta Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2016-06-29 Classification: DNA BINDING PROTEIN Ligands: 67S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 67S
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Identification Of Spirooxindole And Dibenzoxazepine Motifs As Potent Mineralocorticoid Receptor Antagonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-03-09 Classification: SIGNALING PROTEIN Ligands: 60R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-09
Ligands: 60R, CL
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The Structure Of The C.Kpn2I Controller Protein
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-03-02 Classification: GENE REGULATION Ligands: GOL |
Organism: Klebsiella pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: GOL
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Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, CL, RX5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: NAG, CL, RX5
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Clinically Useful Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2011-11-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, RX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-30
Ligands: CL, RX6
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Alkyl Amine Renin Inhibitors: Filling S1 From S3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-08-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: RX0, GOL, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-03
Ligands: RX0, GOL, NAG
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Optimization Of Orally Bioavailable Alkyl Amine Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-01-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 22X, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: 22X, NAG
