Search Count: 11
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Crystal Structure Of Nlrp3 In Complex With Inhibitor Np3-253
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-12-11 Classification: IMMUNE SYSTEM Ligands: A1IPJ, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-11
Ligands: A1IPJ, ADP
 |
Crystal Structure Of Nlrp3 Nacht Domain In Complex With A Potent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2021-10-20 Classification: IMMUNE SYSTEM Ligands: RM5, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-20
Ligands: RM5, ADP
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Rorgt (264-518;C455S) In Complex With The Fragment ("Cpd-1") And Rip140 Peptide At 1.80A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EE8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EE8
 |
Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-2" And Rip140 Peptide At 1.90A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EF5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EF5
 |
Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-9" And Rip140 Peptide At 1.66A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EEZ
 |
Synthesis And Biological Evaluation Of New Triazolo And Imidazolopyridine Rorgt Inverse Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2016-12-14 Classification: TRANSCRIPTION Ligands: Q6Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: Q6Y
 |
Discovery Of Imidazoquinolines As A Novel Class Of Potent, Selective And In Vivo Efficacious Cot Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-08-24 Classification: TRANSFERASE Ligands: 6DA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: 6DA
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(2-Amino-5-(Quinolin-3-Yl)Pyridin-3-Yl)-1,3,4-Oxadiazole-2(3H)-Thione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 49B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 49B
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(5-(1H-Indol-3-Yl)-1H-Pyrrolo[2,3-B]Pyridin-3-Yl)-1,3,4-Oxadiazol-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 499 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 499
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Crystal Structure Analysis Of A 6-Amino Quinazolinedione Sulfonamide Bound To Human Glur2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-01-11 Classification: TRANSPORT PROTEIN/ANTAGONIST Ligands: 08W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: 08W
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Crystal Structure Analysis Of A Quinazolinedione Sulfonamide Bound To Human Glur2: A Novel Class Of Competitive Ampa Receptor Antagonists With Oral Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-05-18 Classification: TRANSPORT PROTEIN Ligands: QSN, GLU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: QSN, GLU