Search Count: 56
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Ask1 Bound To Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2024-07-17 Classification: TRANSFERASE/INHIBITOR Ligands: A1AWT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-17
Ligands: A1AWT
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The Crystal Structure Of A Helical Domain Deleted Parp1 In Complex With Isoindolinone Based Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.02 Å Release Date: 2024-03-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VHU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-27
Ligands: VHU
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Bio-2895 (Brd0705) Bound Gsk3Alpha-Axin Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2023-06-14 Classification: HYDROLASE Ligands: 6VL, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: 6VL, CA
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Bio-8546 Bound Gsk3Alpha-Axin Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-06-14 Classification: HYDROLASE Ligands: D1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: D1E
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Bio-8546 Bound Gsk3Beta-Axin Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2023-06-14 Classification: HYDROLASE Ligands: D1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: D1E
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Bio-2895 (Brd0705) Bound Gsk3Beta-Axin Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-06-14 Classification: HYDROLASE Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: 6VL
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Bruton'S Tyrosine Kinase In Complex With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: ZB9, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: ZB9, DMS, PEG
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Bruton'S Tyrosine Kinase In Complex With An Orthosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-03-01 Classification: TRANSFERASE/INHIBITOR Ligands: DMS, Y8C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: DMS, Y8C
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Bruton'S Tyrosine Kinase In Complex With An Orthosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-03-01 Classification: TRANSFERASE/INHIBITOR Ligands: DMS, Y8H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: DMS, Y8H
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Bruton'S Tyrosine Kinase In Complex With Compound 45
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B9
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Bruton'S Tyrosine Kinase In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0BG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0BG, DMS
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Bruton'S Tyrosine Kinase In Complex With Compound 65
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B0
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Crystal Structure Of Bio-32546 Bound Mouse Autotaxin
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-04-13 Classification: HYDROLASE/INHIBITOR Ligands: ZF7, IOD, EDO, ZN, PEG |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-04-13
Ligands: ZF7, IOD, EDO, ZN, PEG
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Structure Of Ttbk1 Kinase Domain In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2021-05-19 Classification: TRANSFERASE/INHIBITOR Ligands: VP7, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: VP7, NA
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Structure Of Ttbk1 Kinase Domain In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2021-05-19 Classification: TRANSFERASE/INHIBITOR Ligands: VSY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: VSY
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Bruton'S Tyrosine Kinase In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2020-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DMS, RQS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: DMS, RQS
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Bruton'S Tyrosine Kinase In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DMS, DTT, S5M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: DMS, DTT, S5M
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Bruton'S Tyrosine Kinase In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2020-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: S9A, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: S9A, DMS
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Adp Bound Ttbk2 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-06-03 Classification: TRANSFERASE Ligands: ADP, PO4, NA, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: ADP, PO4, NA, MG, GOL
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Structure Of Ask1 Bound To Bio-1772961
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2020-05-06 Classification: TRANSFERASE Ligands: DMS, RFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: DMS, RFG
