Search Count: 52
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Bruton'S Tyrosine Kinase In Complex With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YD7, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: YD7, DMS
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Bruton'S Tyrosine Kinase In Complex With Compound 51
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YDA, DTT, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: YDA, DTT, ACT
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Structure Of Tubulin Tyrosine Ligase In Complex With Tb111
Organism: Rattus norvegicus, Gallus gallus, Sus scrofa
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2021-03-31 Classification: LIGASE Ligands: GTP, MG, CA, GDP, MES, O9B, O9H, OH5, PGE, VAL, ACP |
Organism: Rattus norvegicus, Gallus gallus, Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2021-03-31
Ligands: GTP, MG, CA, GDP, MES, O9B, O9H, OH5, PGE, VAL, ACP
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Structure Of Tubulin Tyrosine Ligase In Complex With Tb116
Organism: Rattus norvegicus, Gallus gallus, Sus scrofa
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2021-03-31 Classification: LIGASE Ligands: GTP, MG, CA, GDP, MES, O9B, O9K, O9N, PGE, VAL, P6S, PEG, ACP |
Organism: Rattus norvegicus, Gallus gallus, Sus scrofa
Method: X-RAY DIFFRACTION
Release Date: 2021-03-31
Ligands: GTP, MG, CA, GDP, MES, O9B, O9K, O9N, PGE, VAL, P6S, PEG, ACP
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Structure Of The Human Jak1 Kinase Domain With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEJ, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEP, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KES, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KES, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: GOL, KEV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: GOL, KEV
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Structure Of The Human Jak1 Kinase Domain With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KEY, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KEY, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 56
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KF1, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KF1, GOL
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Structure Of The Human Jak1 Kinase Domain With Compound 54
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2019-04-24 Classification: IMMUNE SYSTEM Ligands: KF4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: KF4, GOL
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Pim1 In Complex With Cpd16 (5-Amino-N-(5-((4R,5R)-4-Amino-5-Fluoroazepan-1-Yl)-1-Methyl-1H-Pyrazol-4-Yl)-2-(2,6-Difluorophenyl)Thiazole-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: GOL, PO4, KUV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: GOL, PO4, KUV
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Dlk In Complex With Compound 10 (5-(1-Isopropyl-5-(3-(Oxetan-3-Yl)-3-Azabicyclo[3.1.0]Hexan-6-Yl)-1H-Pyrazol-3-Yl)-3-(Trifluoromethyl)Pyridin-2-Amine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2017-10-04 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: 9FS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: 9FS
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Dlk In Complex With Inhibitor 5-(1-Isopropyl-5-(1-(Oxetan-3-Yl)Piperidin-4-Yl)-1H-Pyrazol-3-Yl)-3-(Trifluoromethyl)Pyridin-2-Amine (Compound 7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2017-10-04 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: 9FV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: 9FV
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Glk Co-Crystal Structure With Aminopyrrolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-10-26 Classification: Transferase/Transferase Inhibitor Ligands: 6G2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-26
Ligands: 6G2
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound G-5555
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59T
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound Frax1036
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59U, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59U, DMS
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Structure Of 4497 Fab Bound To Synthetic Wall Teichoic Acid Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2015-11-11 Classification: IMMUNE SYSTEM Ligands: CA, 57S, ACT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: CA, 57S, ACT, GOL
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Discovery Of 3,5-Substituted 6-Azaindazoles As Potent Pan-Pim Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-10-28 Classification: Transferase/Transferase Inhibitor Ligands: L20, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: L20, PO4
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Pim1 In Complex With Cpd4 (3-Methyl-5-(Pyridin-3-Yl)-1H-Pyrazolo[3,4-C]Pyridine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2015-10-28 Classification: Transferase/Transferase Inhibitor Ligands: 5E5, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 5E5, PO4
