Search Count: 6
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi098
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2016-04-20 Classification: TRANSFERASE Ligands: 986, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 986, EDO
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Crystal Structure Of The Cbp Bromodomain In Complex With Cpi703
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING Ligands: 58N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 58N
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Discovery Of Benzotriazolo Diazepines As Orally-Active Inhibitors Of Bet Bromodomains: Crystal Structure Of Brd4 With Cpi-13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2015-11-11 Classification: SIGNALING PROTEIN Ligands: FMT, 3X0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: FMT, 3X0
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Crystal Structure Of The First Bromodomain Of Human Brd4 Bound To Benzotriazolo-Diazepine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2015-04-08 Classification: TRANSCRIPTION Ligands: 558 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 558
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Crystal Structure Of The First Bromodomain Of Human Brd4 With Benzotriazolo-Diazepine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2015-04-08 Classification: SIGNALING PROTEIN Ligands: 559 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 559
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Ibet Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-11-17 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: EAM, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-17
Ligands: EAM, EDO
