Search Count: 29
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Crystal Structure Of The Mycobacterium Tuberculosis Transcriptional Repressor Ethr2 In Complex With Bdm41420
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-04-26 Classification: TRANSCRIPTION Ligands: 69Y |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: 69Y
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Iodinated Form Of The Mycobacterium Tuberculosis Repressor Ethr2
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-04-26 Classification: DNA BINDING PROTEIN Ligands: IOD |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
Ligands: IOD
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Unliganded Form Of The Mycobacterium Tuberculosis Repressor Ethr2
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-04-26 Classification: DNA BINDING PROTEIN |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2017-04-26
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3.1 A Resolution Crystal Structure Of The B. Pertussis Bvgs Periplasmic Domain
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-02-11 Classification: TRANSFERASE |
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
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Novel N-Phenyl-Phenoxyacetamide Derivatives As Potential Ethr Inhibitors And Ethionamide Boosters. Discovery And Optimization Using High-Throughput Synthesis.
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-03-27 Classification: TRANSCRIPTION/INHIBITOR Ligands: 0MN, NH4, GOL |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: 0MN, NH4, GOL
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm31379
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-01-11 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: LL3 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: LL3
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm31369
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2012-01-11 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: LL4 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2012-01-11
Ligands: LL4
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G106W Mutant Of Ethr From Mycobacterium Tuberculosis
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-12-28 Classification: TRANSCRIPTION |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-28
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm33066
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2011-12-21 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: LL5, GOL |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: LL5, GOL
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Structural Activation Of The Transcriptional Repressor Ethr From M. Tuberculosis By Single Amino-Acid Change Mimicking Natural And Synthetic Ligands
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-12-21 Classification: TRANSCRIPTION/INHIBITOR Ligands: FO5 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: FO5
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Structure Of Hth-Type Transcriptional Regulator Ethr, G106W Mutant
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2011-12-21 Classification: TRANSCRIPTION |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
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Ethionamide Boosters Part 2: Combining Bioisosteric Replacement And Structure-Based Drug Design To Solve Pharmacokinetic Issues In A Series Of Potent 1,2,4-Oxadiazole Ethr Inhibitors.
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2011-12-07 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 3SE |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: 3SE
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Ethionamide Boosters Part 2: Combining Bioisosteric Replacement And Structure-Based Drug Design To Solve Pharmacokinetic Issues In A Series Of Potent 1,2,4-Oxadiazole Ethr Inhibitors.
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2011-12-07 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: 3SF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: 3SF
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Crystal Structure Of The R450A Mutant Of The Membrane Protein Fhac
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2010-11-03 Classification: PROTEIN TRANSPORT |
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION
Release Date: 2010-11-03
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Crystal Structure Of Bordetella Pertussis Bvgs Periplasmic Vft2 Domain
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2010-10-06 Classification: SIGNALING PROTEIN Ligands: GOL, ACT |
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: GOL, ACT
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Crystal Structure Of Bordetella Pertussis Bvgs Vft2 Domain (Double Mutant F375E/Q461E)
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-10-06 Classification: SIGNALING PROTEIN Ligands: EDO |
Organism: Bordetella pertussis
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: EDO
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm14801
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-09-01 Classification: TRANSCRIPTION REPRESSOR/INHIBITOR Ligands: O8G |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2010-09-01
Ligands: O8G
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm14950
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-09-01 Classification: TRANSCRIPTION Ligands: O8H |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2010-09-01
Ligands: O8H
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm14744
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2009-07-21 Classification: TRANSCRIPTION Ligands: RF2 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2009-07-21
Ligands: RF2
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Ethr From Mycobacterium Tuberculosis In Complex With Compound Bdm31381
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2009-07-21 Classification: TRANSCRIPTION Ligands: RF3 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2009-07-21
Ligands: RF3
