Search Count: 16
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Pi3K Alpha Lipid Kinase With Active Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-06-17 Classification: Transferase/Transferase Inhibitor Ligands: 4EL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: 4EL
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Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk147
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3YZ
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Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk199
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.29 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3Z0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3Z0
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 11C [N-{2-[1-(6-Carbamoylthieno[3,2-D]Pyrimidin-4-Yl)Piperidin-4-Yl]Ethyl}-N'-Ethylthiophene-2,5-Dicarboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NQ
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 28 [4-(4-{2-[(2,2-Dimethylpropanoyl)Amino]Ethyl}Piperidin-1-Yl)Thieno[3,2-D]Pyrimidine-6-Carboxamide[
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NR
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 3 [14-(4-{2-[(Methylsulfonyl)Amino]Ethyl}Piperidin-1-Yl)Thieno[3,2-D]Pyrimidine-6-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NS, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NS, GOL, NA
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Crystal Structure Of An Extender (Spd28345)-Modified Human Pdk1 Complex 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: SYP
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Pdk1 In Complex With Dfg-Out Inhibitor Xxx
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MP7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: MP7
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-(1-Benzyl-Piperidin-4-Yl)-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1H
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(2,6-Dimethoxy-Benzyl)-Piperidin-4-Yl]-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1I
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With 4-(4-Fluoro-Benzyl)-Piperazine-2-Carboxylic Acid (2-Mercapto-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1J
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With 4-(4-Fluoro-Benzyl)-Piperazine-2-Carboxylic Acid(3-Mercapto-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1K
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Bromo-2,3-Dimethoxy-Benzyl)-Piperidin-4-Yl]-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1L
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Chloro-2-Isopropoxy-3-Methoxy-Benzyl)-Piperidin-4-Yl]-2-(4-Sulfamoyl-Phenoxy)-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1M
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(5-Chloro-2-Isopropoxy-3-Methoxy-Benzyl)-Piperidin-4-Yl]-2-(2-Methyl-4-Sulfamoyl-Phenoxy)-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1N
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Structure Of Tar Rna Complexed With A Tat-Tar Interaction Nanomolar Inhibitor That Was Identified By Computational Screening
Organism: Human immunodeficiency virus 1
Method: SOLUTION NMR Release Date: 2002-12-11 Classification: RNA Ligands: PMZ |
Organism: Human immunodeficiency virus 1
Method: SOLUTION NMR
Release Date: 2002-12-11
Ligands: PMZ