Search Count: 23
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Crystal Structure Of The Human Ttk In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-05-15 Classification: SIGNALING PROTEIN Ligands: KE7, 1PE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: KE7, 1PE, EDO
 |
Ttk In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-10-25 Classification: SIGNALING PROTEIN Ligands: CQ7, CAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-25
Ligands: CQ7, CAC
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y4
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y8
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Discovery Of Novel, Orally Efficacious Liver X Receptor (Lxr) Beta Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2016-06-29 Classification: DNA BINDING PROTEIN Ligands: 67S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 67S
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Identification Of Spirooxindole And Dibenzoxazepine Motifs As Potent Mineralocorticoid Receptor Antagonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-03-09 Classification: SIGNALING PROTEIN Ligands: 60R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-09
Ligands: 60R, CL
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Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With Bms-809959 Aka 4-Tert-Butyl-N-[2-Me Thyl-3-(6-{[4-(Morpholine-4-Carbonyl)Phenyl]Amino}-9H- Purin-2-Yl)Phenyl]Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2P5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2P5
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Crystal Structure Of Mitogen-Activated Protein Kinase 14 (P38-H5) Complex With 5-(2-Chlorophenyl)-N-(5-(Cyclopropylcarbamoyl)-2-Methylphenyl)-2-Thiophenecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2013-06-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1M8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-12
Ligands: 1M8
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Crystal Structure Of Mitogen-Activated Protein Kinase 14 (P38-H5) Complex With 2-(2-Chlorophenyl)-N-(5-(Cyclopropylcarbamoyl)-2-Methylphenyl)-1,3-Thiazole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2013-06-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1R9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-12
Ligands: 1R9
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Crystal Structure Of Mitogen-Activated Protein Kinase 14 (P38-H5) Complex With Ethyl 6-((5-(Cyclopropylcarbamoyl)-2-Methylphenyl)Carbamoyl)-1H-Indole-1-Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-06-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1RA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-12
Ligands: 1RA
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P38 Alpha Kinase Complexed With A Pyrazolo-Triazine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: NK0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: NK0
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P38 Alpha Kinase Complexed With A 5-Amino-Pyrazole Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2010-11-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OCG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-17
Ligands: OCG
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: 38P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 38P
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P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7V
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-10-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 39P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 39P
 |
P38 Alpha Kinase Complexed With A 2-Aminothiazol-5-Yl-Pyrimidine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2010-09-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3NW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: 3NW
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P38 Alpha Kinase Complexed With A Pyrazolo-Pyrimidine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-03-02 Classification: TRANSFERASE Ligands: N4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: N4D
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Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2008-04-15 Classification: TRANSFERASE Ligands: P39 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: P39
 |
P38 Alpha Map Kinase Complexed With Bms-640994
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-15 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: 304 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: 304
 |
Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-08 Classification: TRANSFERASE Ligands: P38 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
Ligands: P38
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P38 Alpha Map Kinase Complexed With A Benzothiazole Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2008-03-25 Classification: TRANSFERASE Ligands: P41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-25
Ligands: P41