Search Count: 41
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Crystal Structure Of Cdk2 Bound By Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1INI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1INI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 11 (Azd8421)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOP
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDP
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDO
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDG
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E3 Ligase Cbl-B In Complex With A Triazolone Core Inhibitor (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEW, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEW, ZN, NA
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E3 Ligase Cbl-B In Complex With A Lactam Scaffold Inhibitor (Compound 7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IEV, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IEV, ZN, NA
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E3 Ligase Cbl-B In Complex With A Carbamate Scaffold Inhibitor (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-07-31 Classification: LIGASE Ligands: A1IE5, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-31
Ligands: A1IE5, ZN, NA
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Bfl1 In Complex With A Reversible Covalent Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2024-07-03 Classification: APOPTOSIS Ligands: A1H2C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: A1H2C
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 31)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-01-24 Classification: LIGASE Ligands: ZN, NA, WX9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-24
Ligands: ZN, NA, WX9
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WUQ, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WUQ, ZN, NA
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: WX0, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: WX0, ZN, NA
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Crystal Structure Of Cbl-B In Complex With An Allosteric Inhibitor (Compound 30)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2024-01-10 Classification: LIGASE Ligands: ZN, NA, WUI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-10
Ligands: ZN, NA, WUI
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Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Benzodiazepine Hts Hit Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: W89, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: W89, ZN, NA
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Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Wo2020264398 Ex23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: Z3N, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: Z3N, ZN, NA
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Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Benzodiazepine Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: W7R, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: W7R, ZN, NA
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Crystal Structure Of D1228V C-Met Bound By Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: GOL, EDO, FMT, W49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: GOL, EDO, FMT, W49
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Crystal Structure Of D1228V C-Met Bound By Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W3R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W3R, CL
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Crystal Structure Of D1228V C-Met Bound By Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2023-07-05 Classification: TRANSFERASE Ligands: W3W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: W3W