Search Count: 30
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Hiv-Rt Pre-Catalytic Complex With Mk-8527
Organism: Hiv-1 m:b_hxb2r, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2025-09-17 Classification: TRANSFERASE/DNA Ligands: MG, A1A6R |
Organism: Hiv-1 m:b_hxb2r, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2025-09-17
Ligands: MG, A1A6R
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Trka With (6~{R})-3-Methylsulfanyl-6-Phenyl-1-(1~{H}-Pyrazol-3-Yl)-6,7-Dihydro-5~{H}-Thieno[3,4-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2017-08-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 69C, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-09
Ligands: 69C, CL, ACT
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Bace1 In Complex With 4-(Cyclohexylamino)-1-(3-Fluorophenyl)-8-(3-Isopropoxybenzyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QA
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Bace1 In Complex With 8-(3-((1-Aminopropan-2-Yl)Oxy)Benzyl)-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4QD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QD
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Bace1 In Complex With 8-Benzyl-4-(Cyclohexylamino)-1-(3-Fluorophenyl)-7-Methyl-1,3,8-Triazaspiro[4.5]Dec-3-En-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-05 Classification: Hydrolase/hydrolase inhibitor Ligands: 4QF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4QF
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The Structure Of Trka Kinase Bound To The Inhibitor N-(3-Cyclopropyl-1-Phenyl-1H-Pyrazol-5-Yl)-2-{4-[3-Methoxy-4-(4-Methyl-1H-Imidazol-1-Yl)Phenyl]-1H-1,2,3-Triazol-1-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31V, GOL, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31V, GOL, CL, ACT
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The Structure Of Trka Kinase Bound To The Inhibitor 1-Cyclopropyl-1-[3-(1,3-Thiazol-2-Yl)Benzyl]-3-[4-(Trifluoromethoxy)Phenyl]Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31W, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31W, CL, ACT
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The Structure Of Trka Kinase Bound To The Inhibitor 4-Naphthalen-1-Yl-1-[(5-Phenyl-1,2,4-Oxadiazol-3-Yl)Methyl]-1H-Pyrrolo[3,2-C]Pyridine-2-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31X, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31X, CL, ACT
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The Structure Of Trka Kinase Bound To The Inhibitor N~4~-(4-Morpholin-4-Ylphenyl)-N~6~-(Pyridin-3-Ylmethyl)Pyrido[3,2-D]Pyrimidine-4,6-Diamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-06-18 Classification: Transferase/Transferase inhibitor Ligands: 31Y, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31Y, CL, ACT
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Crystal Structure Of Hiv-1 Reverse Transcriptase (Wild Type) In Complex With Inhibitor M05
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5MA |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 5MA
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Crystal Structure Of Hiv-1 Reverse Transcriptase (K103N Mutant) In Complex With Inhibitor M05
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-10-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5MA |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: 5MA
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Crystal Structure Of Hiv-1 Reverse Transcriptase (K103N Mutant) In Complex With Inhibitor M06
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2011-10-26 Classification: Transferase/transferase Inhibitor Ligands: M06 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: M06
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Crystal Structure Of Hiv Reverse Transcriptase In Complex With Inhibitor 3
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2009-08-25 Classification: TRANSFERASE Ligands: RT3 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: RT3
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Crystal Structure Of Hiv Reverse Transcriptase In Complex With Inhibitor 7
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-08-25 Classification: TRANSFERASE Ligands: RT7 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2009-08-25
Ligands: RT7
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Discovery Of Aminoheterocycles As A Novel Beta-Secretase Inhibitor Class
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2009-07-07 Classification: HYDROLASE Ligands: B35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-07
Ligands: B35
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Hiv Reverse Transcriptase In Complex With Inhibitor R8E
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-10-14 Classification: TRANSFERASE Ligands: R8E |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: R8E
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Hiv Reverse Transcriptase Y181C Mutant In Complex With Inhibitor R8E
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2008-10-14 Classification: TRANSFERASE Ligands: R8E |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: R8E
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Hiv Reverse Transcriptase K103N Mutant In Complex With Inhibitor R8D
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2008-10-14 Classification: TRANSFERASE Ligands: R8D |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: R8D
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Crystal Structure Of Human Beta Secretase Complexed With Ixs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-04-22 Classification: HYDROLASE Ligands: IXS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: IXS
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Crystal Structure Of Hiv Reverse Transcriptase In Complex With Inhibitor 14
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2008-04-22 Classification: TRANSFERASE Ligands: M14 |
Organism: Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: M14