Search Count: 18
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Factor Xa Complex With Gtc000401
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-09-30 Classification: HYDROLASE Ligands: CA, 4O1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: CA, 4O1
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Factor Xa Complex With Gtc000406
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-09-30 Classification: HYDROLASE Ligands: CA, MG, 4O6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: CA, MG, 4O6
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The Discovery Of Potent And Long-Acting Oral Factor Xa Inhibitors With Tetrahydroisoquinoline And Benzazepine P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-03-16 Classification: BLOOD CLOTTING Ligands: MZA, CA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-16
Ligands: MZA, CA, MG
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Structure And Property Based Design Of Factor Xa Inhibitors: Pyrrolidin-2-Ones With Aminoindane And Phenylpyrrolidine P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2011-03-16 Classification: BLOOD CLOTTING Ligands: C0Z, CA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-16
Ligands: C0Z, CA, MG
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Structure And Property Based Design Of Factor Xa Inhibitors: Pyrrolidin-2-Ones With Aminoindane And Phenylpyrrolidine P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-03-16 Classification: BLOOD CLOTTING Ligands: 439, CA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-16
Ligands: 439, CA, MG
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Structure And Property Based Design Of Factor Xa Inhibitors: Pyrrolidin-2-Ones With Aminoindane And Phenylpyrrolidine P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-03-16 Classification: BLOOD CLOTTING Ligands: 931, CA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-16
Ligands: 931, CA, MG
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Structure And Property Based Design Of Factor Xa Inhibitors: Pyrrolidin-2-Ones With Aminoindane And Phenylpyrrolidine P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-03-16 Classification: BLOOD CLOTTING Ligands: 930, CA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-16
Ligands: 930, CA, MG
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Structure And Property Based Design Of Factor Xa Inhibitors: Pyrrolidin-2-Ones With Monoaryl P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2010-12-01 Classification: BLOOD CLOTTING Ligands: 461 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: 461
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Structure And Property Based Design Of Factor Xa Inhibitors: Pyrrolidin-2-Ones With Monoaryl P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2010-12-01 Classification: BLOOD CLOTTING Ligands: 898 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: 898
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Structure And Property Based Design Of Factor Xa Inhibitors: Pyrrolidin-2-Ones With Biaryl P4 Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2008-12-16 Classification: HYDROLASE Ligands: GSV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-16
Ligands: GSV
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Structure And Property Based Design Of Factor Xa Inhibitors:Biaryl Pyrrolidin-2-Ones Incorporating Basic Heterocyclic Motifs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2008-11-25 Classification: HYDROLASE Ligands: CA, MG, GSI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-25
Ligands: CA, MG, GSI
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Selective And Dual Action Orally Active Inhibitors Of Thrombin And Factor Xa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2007-05-08 Classification: HYDROLASE Ligands: 701 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-05-08
Ligands: 701
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Factor Xa Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2007-05-08 Classification: HYDROLASE Ligands: 894, CA, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-05-08
Ligands: 894, CA, MG
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Selective And Dual Action Orally Active Inhibitors Of Thrombin And Factor Xa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2007-04-24 Classification: HYDROLASE Ligands: 895 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-04-24
Ligands: 895
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Crystal Structure Of A Human Factor Xa Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-03-20 Classification: HYDROLASE Ligands: G15, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: G15, CA
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Crystal Structure Of A Human Factor Xa Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2007-03-20 Classification: HYDROLASE Ligands: GSX, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-03-20
Ligands: GSX, CA
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Crystal Structure Of A Human Factor Xa Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2006-09-27 Classification: HYDROLASE Ligands: GSJ, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-09-27
Ligands: GSJ, CA
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Crystal Structure Of A Human Factor Xa Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2006-05-17 Classification: HYDROLASE Ligands: CA, GSK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-05-17
Ligands: CA, GSK
