Search Count: 28
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Pitp In Complex With The Inhibitor Vt01545
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2024-05-08 Classification: LIPID BINDING PROTEIN Ligands: IMD, GOL, NI |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-05-08
Ligands: IMD, GOL, NI
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Crystal Structure Of Tead3 In Complex With Vt105
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-04-28 Classification: DNA BINDING PROTEIN Ligands: G9O, PO4, CL, G9C, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-28
Ligands: G9O, PO4, CL, G9C, TRS
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Co-Crystal Structure Of P. Aeruginosa Lpxc-50067 Complex
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: MG, JWM |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: MG, JWM
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Co-Crystal Structure Of P. Aeruginosa Lpxc-50228 Complex
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: JWP, MG |
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Co-Crystal Structure Of P. Aeruginosa Lpxc-50432 Complex
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: MG, JWV, GOL |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: MG, JWV, GOL
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Co-Crystal Structure Of P. Aeruginosa Lpxc-Achn975 Complex
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: ZN, A5F |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: ZN, A5F
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Crystal Structures Of Apo Keap1, Keap1-Peptide, And Keap1-Compound Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-08-20 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-20
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R78 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: R78
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1D1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: 1D1
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Crystal Structures Of Apo Keap1, Keap1-Peptide, And Keap1-Compound Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-12-18 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
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Crystal Structures Of Apo Keap1, Keap1-Peptide, And Keap1-Compound Complexes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-12-18 Classification: TRANSCRIPTION Ligands: 12O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: 12O
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-11-20 Classification: transferase/transferase inhibitor Ligands: 11G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 11G
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce -Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-11-20 Classification: transferase/transferase inhibitor Ligands: 1C7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 1C7
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Selective & Brain-Permeable Polo-Like Kinase-2 (Plk-2) Inhibitors That Reduce Alpha-Synuclein Phosphorylation In Rat Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-08-14 Classification: transferase/transferase inhibitor Ligands: 1C8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1C8
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Design And Synthesis Of Brain Penetrant Selective Jnk Inhibitors With Improved Pharmacokinetic Properties For The Prevention Of Neurodegeneration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-05-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 34I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-08
Ligands: 34I
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 0ZA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 0ZA
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1B9
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: 1BB, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: 1BB, ZN
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1BS
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2013-03-06 Classification: transferase/transferase inhibitor Ligands: ZN, 1CH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1CH