Search Count: 14
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Bace1 Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2018-04-18 Classification: PEPTIDE BINDING PROTEIN Ligands: B7E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: B7E
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Bace1 Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2018-04-18 Classification: PEPTIDE BINDING PROTEIN Ligands: B7T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-18
Ligands: B7T
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Lead Generation Of Bace1 Inhibitors By Coupling Non-Amidine New Warheads To A Known Binding Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2013-07-24 Classification: HYDROLASE Ligands: GMF, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-24
Ligands: GMF, ACT
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Design And Synthesis Of Bace1 Inhibitors With In Vivo Brain Reduction Of Beta-Amyloid Peptides (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2012-10-17 Classification: HYDROLASE Ligands: ACT, NA, 7F3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-17
Ligands: ACT, NA, 7F3
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Design And Synthesis Of Bace1 Inhibitors With In Vivo Brain Reduction Of Beta-Amyloid Peptides (Compound (R)-41)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2012-10-17 Classification: HYDROLASE Ligands: ACT, I6X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-17
Ligands: ACT, I6X
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Preclinical Characterization Of Azd3839, A Novel Clinical Candidate Bace1 Inhibitor For The Treatment Of Alzheimer Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-10-17 Classification: HYDROLASE Ligands: ACT, NA, 32D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-17
Ligands: ACT, NA, 32D
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New Aminoimidazoles As Bace-1 Inhibitors: From Rational Design To Ab- Lowering In Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2012-10-10 Classification: HYDROLASE Ligands: DMS, 1B1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: DMS, 1B1
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New Aminoimidazoles As Bace-1 Inhibitors: From Rational Design To Ab- Lowering In Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2012-10-10 Classification: HYDROLASE Ligands: ACT, 6TG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: ACT, 6TG
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New Aminoimidazoles As Bace-1 Inhibitors: From Rational Design To Ab- Lowering In Brain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2012-10-10 Classification: HYDROLASE Ligands: 6T6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 6T6
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Aminoimidazoles As Bace-1 Inhibitors. X-Ray Crystal Structure Of Beta Secretase Complexed With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2012-02-29 Classification: HYDROLASE Ligands: ACT, QN7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-29
Ligands: ACT, QN7
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Aminoimidazoles As Bace-1 Inhibitors. X-Ray Crystal Structure Of Beta Secretase Complexed With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-02-29 Classification: HYDROLASE Ligands: ACT, S8Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-29
Ligands: ACT, S8Z
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X-Ray Crystal Structure Of Beta Secretase Complexed With Compound 8C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2007-11-13 Classification: HYDROLASE Ligands: IOD, C8C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-13
Ligands: IOD, C8C
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X-Ray Crystal Structure Of Beta Secretase Complexed With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-11-13 Classification: HYDROLASE Ligands: IOD, H24 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-13
Ligands: IOD, H24
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X-Ray Crystal Structure Of Beta Secretase Complexed With Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-11-13 Classification: HYDROLASE Ligands: IOD, C27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-13
Ligands: IOD, C27
