Search Count: 30
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Kras G12D In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2024-10-02 Classification: ONCOPROTEIN Ligands: GCP, YLE, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GCP, YLE, MG
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Kras G12D In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2024-10-02 Classification: ONCOPROTEIN Ligands: GCP, MG, YFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GCP, MG, YFJ
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Protac-Mediated Complex Of Kras With Vhl/Elongin-B/Elongin-C/Cullin-2/Rbx1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.50 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: ZN, GDP, WYL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-12-06
Ligands: ZN, GDP, WYL
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Kras-G12C In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: GDP, MG, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, MG, WYU
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Crystal Structure Of Ligand Acbi3 In Complex With Kras G12D C118S Gdp And Pvhl:Elonginc:Elonginb Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2023-12-06 Classification: GENE REGULATION Ligands: PO4, WYL, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: PO4, WYL, GDP, MG
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Crystal Structure Of Compound 3 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: GDP, X4R, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, X4R, MG
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Crystal Structure Of Compound 4 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: X53, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: X53, GDP, MG
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Crystal Structure Of Compound 10 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IOD, IFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IOD, IFJ
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Crystal Structure Of Compound 6 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IFF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IFF
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Crystal Structure Of Compound 4 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IF8, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IF8, ZN
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Crystal Structure Of Protac 5 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2022-09-07 Classification: LIGASE Ligands: IEI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-07
Ligands: IEI
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Crystal Structure Of Crystal Form 2 Of An Active Kras G12D (Gppcp) Dimer In Complex With Bi-5747
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2020-11-18 Classification: SIGNALING PROTEIN Ligands: MG, GCP, R6W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: MG, GCP, R6W
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: GCP, MG, F0N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GCP, MG, F0N
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: MG, NO3, GCP, EZZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: MG, NO3, GCP, EZZ
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: MG, GCP, F0B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: MG, GCP, F0B
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Crystal Structure Of Kras G12D (Gppcp) In Complex With Bi 2852
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: F0K, MG, GCP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: F0K, MG, GCP
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Crystal Structure Of Protac 2 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-06-12 Classification: GENE REGULATION Ligands: EDO, FWZ, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: EDO, FWZ, EPE
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Crystal Structure Of Protac 1 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2019-06-12 Classification: GENE REGULATION Ligands: FX8, EDO, FMT, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: FX8, EDO, FMT, EPE
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Crystal Structure Of The Bromodomain Of Human Smarca2 In Complex With Smarca-Bd Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2019-06-12 Classification: GENE REGULATION Ligands: FX5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: FX5, ZN
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Crystal Structure Of Protac 2 In Complex With The Bromodomain Of Human Smarca4 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-06-12 Classification: TRANSCRIPTION Ligands: FWZ, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: FWZ, DMS, EDO
