Search Count: 16
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Catalytic Unit Of Pi3Kg In Complex With Pi3K/Mtor Dual Inhibitor Pf-04979064
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-11-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 19P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: 19P
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Design And Synthesis Of A Novel Pyrrolidinyl Pyrido Pyrimidinone Derivative As A Potent Inhibitor Of Pi3Ka And Mtor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-04-03 Classification: Transferase/Transferase Inhibitor Ligands: 0TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-03
Ligands: 0TA
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Design And Synthesis Of A Novel Pyrrolidinyl Pyrido Pyrimidinone Derivative As A Potent Inhibitor Of Pi3Ka And Mtor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-04-03 Classification: Transferase/Transferase Inhibitor Ligands: 0TB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-03
Ligands: 0TB
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Crystal Structure Of The Human P21-Activated Kinase 4 In Complex With (S)-N-(5-(3-Benzyl-1-Methylpiperazine-4-Carbonyl)-6,6-Dimethyl-1,4,5, 6-Tetrahydropyrrolo(3,4-C)Pyrazol-3-Yl)-3-Phenoxybenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-06-06 Classification: TRANSFERASE Ligands: N53, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-06
Ligands: N53, GOL
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Quinazolines With Intra-Molecular Hydrogen Bonding Scaffold (Imhbs) As Pi3K/Mtor Dual Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2011-02-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3RE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: 3RE
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Quinazolines With Intra-Molecular Hydrogen Bonding Scaffold (Imhbs) As Pi3K/Mtor Dual Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-02-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3RZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: 3RZ
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Quinazolines With Intra-Molecular Hydrogen Bonding Scaffold (Imhbs) As Pi3K/Mtor Dual Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-02-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3PS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: 3PS
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4-Methylpteridineones As Orally Active And Selective Pi3K/Mtor Dual Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2010-09-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OAW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-22
Ligands: OAW
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Discovery Of The Highly Potent Pi3K/Mtor Dual Inhibitor Pf-04691502 Through Structure Based Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-06-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ML8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: ML8
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Discovery Of The Highly Potent Pi3K/Mtor Dual Inhibitor Pf-04691502 Through Structure Based Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2010-06-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ML9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: ML9
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Crystal Structure Of The Human P21-Activated Kinase 4 In Complex With Pf-03758309
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-05-19 Classification: TRANSFERASE Ligands: GOL, 7KC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-05-19
Ligands: GOL, 7KC
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Human Calcineurin Heterodimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 1997-12-03 Classification: HYDROLASE Ligands: ZN, FE, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1997-12-03
Ligands: ZN, FE, CA
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Crystal Structures Of The Myristylated Catalytic Subunit Of Camp-Dependent Protein Kinase Reveal Open And Closed Conformations
Organism: Sus scrofa, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 1994-05-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MYR, IOD |
Organism: Sus scrofa, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-05-31
Ligands: MYR, IOD
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2.0 Angstrom Refined Crystal Structure Of The Catalytic Subunit Of Camp-Dependent Protein Kinase Complexed With A Peptide Inhibitor And Detergent
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1993-04-15 Classification: TRANSFERASE(PHOSPHOTRANSFERASE) Ligands: OCT |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1993-04-15
Ligands: OCT
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2.2 Angstrom Refined Crystal Structure Of The Catalytic Subunit Of Camp-Dependent Protein Kinase Complexed With Mnatp And A Peptide Inhibitor
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1993-04-15 Classification: TRANSFERASE(PHOSPHOTRANSFERASE) Ligands: MN, ATP |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1993-04-15
Ligands: MN, ATP
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Crystal Structure Of The Catalytic Subunit Of Cyclic Adenosine Monophosphate-Dependent Protein Kinase
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 1993-01-15 Classification: TRANSFERASE(PHOSPHOTRANSFERASE) |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 1993-01-15