Search Count: 7
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Crystal Structure Of Plk1 In Complex With A Novel 5,6-Dihydroimidazolo[1,5-F]Pteridine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: 79D, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 79D, ZN
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Crystal Structure Of Plk1 In Complex With A Novel 5,6-Dihydroimidazolo[1,5-F]Pteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: ZN, 79C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 79C
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Structure-Based Optimization Of 1H-Imidazole-2-Carboxamides As Axl Kinase Inhibitors Utilizing A Mer Mutant Surrogate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2017-01-25 Classification: Transferase/Transferase Inhibitor Ligands: 79Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 79Y
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Structure-Based Optimization Of 1H-Imidazole-2-Carboxamides As Axl Kinase Inhibitors Utilizing A Mer Mutant Surrogate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2017-01-25 Classification: Transferase/Transferase Inhibitor Ligands: 7AE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 7AE
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Parp Complexed With Benzo[1,4]Oxazin-3-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-08-07 Classification: transferase/transferase inhibitor Ligands: 1WQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: 1WQ
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Crystal Structure Of Plk1 In Complex With A Pyrimidodiazepinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J3, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 1J3, ZN, ACT
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Crystal Structure Of Plk1 In Complex With Tak-960
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, ACT, 1J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: ZN, ACT, 1J4
