Search Count: 11
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Crystal Structure Of Cyp46A1 With [(1R,5S)-3-Oxa-8-Azabicyclo[3.2.1]Octan-8-Yl][(4R,8M)-8-(1,3-Oxazol-5-Yl)-6-(Trifluoromethyl)Imidazo[1,2-A]Pyridin-3-Yl]Methanone (Compound 3K)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2025-07-02 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-02
Ligands: HEM, A1BZE
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Crystal Structure Of Cyp46A1 With (Morpholin-4-Yl)[(4R,8M)-8-(1,3-Oxazol-5-Yl)-6-(Trifluoromethyl)Imidazo[1,2-A]Pyridin-3-Yl]Methanone (Compound 2H)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2025-07-02 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-02
Ligands: HEM, A1BZD
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Crystal Structure Of Cyp46A1 With Cyclopropyl[(4M)-4-(1,3-Oxazol-5-Yl)-6-(Trifluoromethyl)-1H-Indol-1-Yl]Methanone (Compound 2B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2025-07-02 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZC, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-02
Ligands: HEM, A1BZC, EDO
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Crystal Structure Of Cyp46A1 With 3-Chloro-N-[(3M)-3-(1,3-Oxazol-5-Yl)Phenyl]-N-(Propan-2-Yl)Benzene-1-Sulfonamide (Compound 2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2025-04-23 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-23
Ligands: HEM, A1BZB, EDO
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Crystal Structure Of Cyp46A1 With 3-Chloro-N-[(3M)-3-(1,3-Oxazol-5-Yl)-5-(Trifluoromethyl)Phenyl]Benzamide (Compound 3F)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2025-04-23 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-23
Ligands: HEM, A1BZA
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Crystal Structure Of Cyp46A1 With N-[6-(1,3-Oxazol-5-Yl)-4-(Trifluoromethyl)Pyridin-2-Yl]Cyclopropanecarboxamide (Compound 4L)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2025-04-23 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BY9, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-23
Ligands: HEM, A1BY9, EDO
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Molecular Mechanism Of The The Wake-Promoting Agent Tak-925
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2022-06-08 Classification: SIGNALING PROTEIN Ligands: A6F, OLA |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2022-06-08
Ligands: A6F, OLA
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Structure Of The Orexin-2 Receptor(Ox2R) Bound To Tak-925, Gi And Scfv16
Organism: Homo sapiens, Bos taurus, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2022-05-25 Classification: MEMBRANE PROTEIN Ligands: OLA, A6F |
Organism: Homo sapiens, Bos taurus, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2022-05-25
Ligands: OLA, A6F
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Gsk3Beta Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-03-02 Classification: TRANSFERASE Ligands: G3B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: G3B
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X-Ray Co-Crystal Structure Of Glycogen Synthase Kinase 3Beta In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-03-10 Classification: TRANSFERASE Ligands: 34O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: 34O
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Glycogen Synthase Kinase 3Beta Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-03-10 Classification: TRANSFERASE Ligands: 3HT, 2HT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: 3HT, 2HT