Search Count: 47
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Crystal Structure Of Selective Ire1A Inhibitor 29 At The Enzyme Active Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, XOE
 |
Cryo-Em Structure Of Mal De Rio Cuarto Virus P9-1 Viroplasm Protein (Decamer)
Organism: Mal de rio cuarto virus
Method: ELECTRON MICROSCOPY Release Date: 2022-06-15 Classification: VIRAL PROTEIN |
Organism: Mal de rio cuarto virus
Method: ELECTRON MICROSCOPY
Release Date: 2022-06-15
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Cryo-Em Structure Of Mal De Rio Cuarto Virus P9-1 Viroplasm Protein (Dodecamer)
Organism: Mal de rio cuarto virus
Method: ELECTRON MICROSCOPY Release Date: 2022-06-15 Classification: VIRAL PROTEIN |
Organism: Mal de rio cuarto virus
Method: ELECTRON MICROSCOPY
Release Date: 2022-06-15
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Crystal Structure Of Ire1A In Complex With G-6904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: N8S, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N8S, EPE
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Crystal Structure Of Ire1 In Complex With G-3053
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-04-21 Classification: TRANSFERASE/INHIBITOR Ligands: N97 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: N97
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Crystal Structure Of Ire1A In Complex With G-4100
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2021-04-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
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Crystal Structure Of Mal De Rio Cuarto Virus P9-1 Viroplasm Protein (C-Arm Deletion Mutant)
Organism: Mal de rio cuarto virus
Method: X-RAY DIFFRACTION Resolution:3.47 Å Release Date: 2021-03-17 Classification: VIRAL PROTEIN |
Organism: Mal de rio cuarto virus
Method: X-RAY DIFFRACTION
Release Date: 2021-03-17
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Ternary Complex Of Vhl/Brd4-Bd1/Compound9 (4-(3,5-Difluoropyridin-2-Yl)-N-(11-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-Methylthiazol-5-Yl)Benzyl)Carbamoyl)Pyrrolidin-1-Yl)-3,3-Dimethyl-1-Oxobutan-2-Yl)Amino)-11-Oxoundecyl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-02-24 Classification: PEPTIDE BINDING PROTEIN Ligands: WEP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEP
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Brd4-Bd1 Compound6 (Methyl 4-(3,5-Difluoropyridin-2-Yl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2021-02-24 Classification: CELL CYCLE Ligands: WEM, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-24
Ligands: WEM, GOL
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Structure Of Unphosphorylated Ire1 In Complex With G-1749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJG
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Structure Of Unphosphorylated Ire1 In Complex With G-7658
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJM
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Structure Of Apo Unphosphorylated Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Apo Ire1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-12-09 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
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Structure Of Phosphorylated Ire1 In Complex With G-0701
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2020-12-09 Classification: TRANSFERASE Ligands: SJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJV
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Structure Of Unphosphorylated Human Ire1 Bound To G-9807
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2020-12-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SJS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: SJS
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Crystal Structure Of Ire1A In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QFV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: QFV, GOL
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Crebbp Bromodomain In Complex With Cpd 4 (1-(1-(Cyclopropylmethyl)-3-(1H-Indol-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-08-08 Classification: PROTEIN BINDING/INHIBITOR Ligands: DMS, EDO, BKD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: DMS, EDO, BKD
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Crebbp Bromodomain In Complex With Cpd3 ((S)-1-(3-(6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9U7
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Crebbp Bromodomain In Complex With Cpd8 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydrofuran-3-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2018-03-07 Classification: TRANSFERASE/INHIBITOR Ligands: 9UA, DMS, GOL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UA, DMS, GOL
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Crebbp Bromodomain In Complex With Cpd10 (1-(3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-03-07 Classification: TRANSCRIPTION REGULATOR/INHIBITOR Ligands: 9UD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 9UD