Search Count: 21
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Indazole Inhibitor Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2024-09-18 Classification: TRANSFERASE Ligands: A1AV4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-18
Ligands: A1AV4, EDO
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Structure Of Compound 2 Bound To The Chk1 10-Point Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2023-11-01 Classification: TRANSFERASE Ligands: ZXH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-01
Ligands: ZXH
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Structure Of Compound 5 Bound To The Chk1 10-Point Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2023-11-01 Classification: TRANSFERASE Ligands: ZXL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-01
Ligands: ZXL
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Structure Of Compound 13 Bound To The Chk1 10-Point Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-11-01 Classification: TRANSFERASE Ligands: ZXP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-01
Ligands: ZXP
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Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2023-02-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: UUF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: UUF
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Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2023-02-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: UU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: UU6
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Human Pi3Kdelta In Complex With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2022-02-16 Classification: TRANSFERASE Ligands: YA7, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-16
Ligands: YA7, CL
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 06
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BVI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BVI, EDO
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 09
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BWI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BWI, EDO
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BXI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BXI
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: L80 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: L80
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BYL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: BYL
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Structure Of Chk1 10-Pt. Mutant Complex With Lrrk2 Inhibitor 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2021-06-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-16
Ligands: YXD
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Human Pi3Kdelta In Complex With Compound 2-10 ((3S)-3-Benzyl-3-Methyl-5-[5-(2-Methylpyrimidin-5-Yl)Pyrazolo[1,5-A]Pyrimidin-3-Yl]-1,3-Dihydro-2H-Indol-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2019-08-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P5J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: P5J
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Human Pi3Kalpha In Complex With Compound 2-10 ((3S)-3-Benzyl-3-Methyl-5-[5-(2-Methylpyrimidin-5-Yl)Pyrazolo[1,5-A]Pyrimidin-3-Yl]-1,3-Dihydro-2H-Indol-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2019-08-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P5J, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: P5J, GOL
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Human Pi3Kdelta In Complex With Compound 4-2 ((3S)-1'-(Cyclopropanecarbonyl)-5-(Quinoxalin-6-Yl)Spiro[Indole-3,2'-Pyrrolidin]-2(1H)-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2019-08-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: P5V
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Murine Pi3K Delta Kinsae Domain - Cpd 1
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: K4A |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: K4A
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Murine Pi3K Delta Kinsae Domain - Cpd 3
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: K47 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: K47
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Crystal Structure Of Sam-Bound Prdm9 In Complex With Mrk-740 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2019-02-13 Classification: GENE REGULATION/INHIBITOR Ligands: ZN, SAM, KS7, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-13
Ligands: ZN, SAM, KS7, UNX
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Irak4 Kinase - Compound 1 Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-05-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 76Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: 76Q
