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Discovery Of Mk-8189, A Highly Potent And Selective Pde10A Inhibitor For The Treatment Of Schizophrenia

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Pde10 Complexed With 5-Chloro-N-[(2,4-Dimethylthiazol-5-Yl)Methyl]Pyrazolo[1,5-A]Pyrimidin-7-Amine

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Pde10 Complexed With N-[(1-Methylpyrazol-4-Yl)Methyl]-5-[[(1S,2S)-2-(2-Pyridyl)Cyclopropyl]Methoxy]Pyrazolo[1,5-A]Pyrimidin-7-Amine
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