Search Count: 18
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Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 5 (1-Methyl-4-Phenylpyrrolidin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: RLG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: RLG
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Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 7B (1-Methyl-4-(4-(Piperidin-1-Ylsulfonyl)Phenyl)Pyrrolidin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: RLS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: RLS
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Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 7H (4-(1-Methyl-5-Oxopyrrolidin-3-Yl)-N-Propylbenzenesulfonamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: RLV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: RLV
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Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 15C (N,N-Diethyl-3',4'-Dimethoxy-6-(1-Methyl-5-Oxopyrrolidin-3-Yl)-[1,1'-Biphenyl]-3-Sulfonamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: NO3, RLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: NO3, RLY
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Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 10 (Methyl [(3R)-1-Methyl-5-Oxopyrrolidin-3-Yl]Acetate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2019-11-27 Classification: PROTEIN BINDING Ligands: OWA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: OWA
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Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 17 (5-{2-[(3R)-1-Methyl-5-Oxopyrrolidin-3-Yl]Ethyl}-2,3,4,5-Tetrahydro-1H-Pyrido[4,3-B]Indol-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.21 Å Release Date: 2019-11-27 Classification: PROTEIN BINDING Ligands: Y17 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: Y17
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Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 18 (5-{[(3R)-1-Methyl-5-Oxopyrrolidin-3-Yl]Methyl}-2,3,4,5-Tetrahydro-1H-Pyrido[4,3-B]Indol-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2019-11-27 Classification: PROTEIN BINDING Ligands: Y18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: Y18
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Induced Myeloid Leukemia Cell Differentiation Protein Fabcomplex In Complex With Azd5991
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-12-26 Classification: APOPTOSIS Ligands: E4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4W
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Mcl1 In Complex With An Indole Acid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-12-26 Classification: IMMUNE SYSTEM Ligands: E4Q, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4Q, EDO
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Mcl1 In Complex With Indole Acid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-12-26 Classification: IMMUNE SYSTEM Ligands: E4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4K
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Crystal Structure Of Myst Acetyltransferase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-08-01 Classification: TRANSFERASE Ligands: CL, ZN, GOL, NA, 7KM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: CL, ZN, GOL, NA, 7KM
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Crystal Structure Of Myst Acetyltransferase Domain In Complex With Acetyl-Coa Cofactor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2018-08-01 Classification: TRANSFERASE Ligands: ZN, NA, ACO, 7L1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: ZN, NA, ACO, 7L1
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Myst Histone Acetyltransferase Kat6A/B In Complex With Wm-1119
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2018-08-01 Classification: TRANSFERASE/INHIBITOR Ligands: FCV, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: FCV, ZN, MG
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Structural Basis Of Cytosolic Dna Recognition By Innate Immune Receptors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2012-04-25 Classification: DNA BINDING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
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Structural Basis Of Cytosolic Dna Recognition By Innate Receptors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-04-25 Classification: DNA BINDING PROTEIN Ligands: EDO, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: EDO, FMT
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Structural Basis Of Cytosolic Dna Recognition By Innate Immune Receptors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2012-04-25 Classification: Immune system/DNA Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: EDO
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Structural Basis Of Cytosolic Dna Recognition By Innate Immune Receptors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-04-25 Classification: Immune system/DNA Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: EDO
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Structural Basis Of Cytosolic Dna Sensing By Innate Immune Receptors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-04-25 Classification: transcription activator/dna Ligands: FMT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: FMT, EDO
