Search Count: 15
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Structure-Based Design Of C8-Substituted O6-Cyclohexylmethoxyguanine Cdk1 And 2 Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2014-12-10 Classification: CELL CYCLE Ligands: 4QE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: 4QE
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Structure-Based Design Of C8-Substituted O6-Cyclohexylmethoxyguanine Cdk1 And 2 Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-12-10 Classification: TRANSFERASE Ligands: 2WC, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: 2WC, MG
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Structure-Based Design Of C8-Substituted O6-Cyclohexylmethoxyguanine Cdk1 And 2 Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-12-10 Classification: TRANSFERASE Ligands: 75X, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: 75X, MG
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Structure-Based Design Of C8-Substituted O6-Cyclohexylmethoxyguanine Cdk1 And 2 Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2014-12-10 Classification: CELL CYCLE Ligands: G6T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: G6T
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Structure-Based Design Of C8-Substituted O6-Cyclohexylmethoxyguanine Cdk1 And 2 Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-12-18 Classification: CELL CYCLE Ligands: JYM, DTT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: JYM, DTT
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Structure-Based Design Of C8-Substituted O6-Cyclohexylmethoxyguanine Cdk1 And 2 Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2013-12-18 Classification: CELL CYCLE Ligands: SQ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-18
Ligands: SQ9
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Co-Crystal Structure Of 6-Cyclohexylmethoxy-8-Isopropyl-9H-Purin-2- Ylamine And Monomeric Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2006-08-30 Classification: TRANSFERASE Ligands: N69 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-08-30
Ligands: N69
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Cdk2 In Complex With A Disubstituted 4, 6-Bis Anilino Pyrimidine Cdk4 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2004-05-04 Classification: TRANSFERASE Ligands: 3FP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-05-04
Ligands: 3FP
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Imidazopyridines: A Potent And Selective Class Of Cyclin-Dependent Kinase Inhibitors Identified Through Structure-Based Hybridisation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2003-09-04 Classification: KINASE Ligands: HDU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-04
Ligands: HDU
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Imidazopyridines: A Potent And Selective Class Of Cyclin-Dependent Kinase Inhibitors Identified Through Structure-Based Hybridisation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2003-09-04 Classification: KINASE Ligands: HDY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-04
Ligands: HDY
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Imidazopyridines: A Potent And Selective Class Of Cyclin-Dependent Kinase Inhibitors Identified Through Structure-Based Hybridisation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2003-09-04 Classification: KINASE Ligands: HDT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-04
Ligands: HDT
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Cdk2 In Complex With A Disubstituted 4, 6-Bis Anilino Pyrimidine Cdk4 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2003-07-11 Classification: TRANSFERASE Ligands: FAP, FCP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-07-11
Ligands: FAP, FCP
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Cdk2 In Complex With A Disubstituted 2, 4-Bis Anilino Pyrimidine Cdk4 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2003-07-11 Classification: TRANSFERASE Ligands: GOL, FAL, FBL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-07-11
Ligands: GOL, FAL, FBL
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Cdk2 In Complex With A Disubstituted 4, 6-Bis Anilino Pyrimidine Cdk4 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2003-07-11 Classification: TRANSFERASE Ligands: MFP, MFQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-07-11
Ligands: MFP, MFQ
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Cdk2 In Complex With A Disubstituted 2, 4-Bis Anilino Pyrimidine Cdk4 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2003-07-11 Classification: TRANSFERASE Ligands: BYP, BWP, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-07-11
Ligands: BYP, BWP, GOL
