Search Count: 7
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Fragment-Based Discovery Of Pyrazolopyridones As Jak1 Inhibitors With Excellent Subtype Selectivity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2020-06-10 Classification: TRANSFERASE Ligands: QZ8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: QZ8
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Fragment-Based Discovery Of Pyrazolopyridones As Jak1 Inhibitors With Excellent Subtype Selectivity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2020-06-10 Classification: TRANSFERASE Ligands: NTW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: NTW
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Fragment-Based Discovery Of Pyrazolopyridones As Jak1 Inhibitors With Excellent Subtype Selectivity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2020-06-10 Classification: TRANSFERASE Ligands: NTQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-10
Ligands: NTQ
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Glucocorticoid Receptor In Complex With Budesonide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-10-04 Classification: SIGNALING PROTEIN Ligands: CPS, EDO, GOL, 8W5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CPS, EDO, GOL, 8W5
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Glucocorticoid Receptor In Complex With Azd5423
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-10-04 Classification: HORMONE Ligands: EDO, 8W8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: EDO, 8W8
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Fragment-Based Discovery Of 6-Arylindazole Jak Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-04-27 Classification: TRANSFERASE Ligands: 6DP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-27
Ligands: 6DP
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The Discovery Of Potent Selective Glucocorticoid Receptor Modulators, Suitable For Inhalation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-05-07 Classification: SIGNALING PROTEIN Ligands: EDO, NN7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: EDO, NN7
