Search Count: 18
![]() |
Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 5 (1-Methyl-4-Phenylpyrrolidin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: RLG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: RLG
![]() |
Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 7B (1-Methyl-4-(4-(Piperidin-1-Ylsulfonyl)Phenyl)Pyrrolidin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: RLS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: RLS
![]() |
Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 7H (4-(1-Methyl-5-Oxopyrrolidin-3-Yl)-N-Propylbenzenesulfonamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: RLV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: RLV
![]() |
Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 15C (N,N-Diethyl-3',4'-Dimethoxy-6-(1-Methyl-5-Oxopyrrolidin-3-Yl)-[1,1'-Biphenyl]-3-Sulfonamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2020-02-26 Classification: PROTEIN BINDING Ligands: NO3, RLY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: NO3, RLY
![]() |
Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 10 (Methyl [(3R)-1-Methyl-5-Oxopyrrolidin-3-Yl]Acetate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2019-11-27 Classification: PROTEIN BINDING Ligands: OWA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: OWA
![]() |
Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 17 (5-{2-[(3R)-1-Methyl-5-Oxopyrrolidin-3-Yl]Ethyl}-2,3,4,5-Tetrahydro-1H-Pyrido[4,3-B]Indol-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.21 Å Release Date: 2019-11-27 Classification: PROTEIN BINDING Ligands: Y17 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: Y17
![]() |
Crystal Structure Of Brd4 Bromodomain 1 With N-Methylpyrrolidin-2-One (Nmp) Derivative 18 (5-{[(3R)-1-Methyl-5-Oxopyrrolidin-3-Yl]Methyl}-2,3,4,5-Tetrahydro-1H-Pyrido[4,3-B]Indol-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2019-11-27 Classification: PROTEIN BINDING Ligands: Y18 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: Y18
![]() |
Crystal Structure Of The Catalytic Domain Of Pde4D2 With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-01-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2SR, EDO, PEG, ZN, DMS, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-21
Ligands: 2SR, EDO, PEG, ZN, DMS, EPE
![]() |
Crystal Structure Of P110Alpha In Complex With Nish2 Of P85Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2014-09-03 Classification: TRANSFERASE/TRANSFERASE REGULATOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
![]() |
Crystal Structure Of Pi3Kalpha In Complex With Dic4-Pip2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2014-09-03 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: PBU, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: PBU, PO4
![]() |
Crystal Structure Of The Apo Form Of The Catalytic Domain Of Pde4D2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-10-26 Classification: HYDROLASE Ligands: EDO, PEG, ZN, PO4, DMS, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: EDO, PEG, ZN, PO4, DMS, EPE
![]() |
Crystal Structure Of The Catalytic Domain Of Pde4D2 With Compound 10D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-10-26 Classification: Hydrolase/Inhibitor Ligands: ZN, EDO, DMS, PEG, PO4, JN4, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: ZN, EDO, DMS, PEG, PO4, JN4, EPE
![]() |
Crystal Structure Of The Catalytic Domain Of Pde4D2 Complexed With Compound 10D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2011-10-26 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, J25, EDO, DMS, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: ZN, J25, EDO, DMS, EPE
![]() |
Crystal Structure Of The Catalytic Domain Of Pde4D2 With Compound 12C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2011-10-26 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, EDO, JN8, DMS, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: ZN, EDO, JN8, DMS, EPE
![]() |
Crystal Structure Of The Catalytic Domain Of Pde4D2 With Compound 10O
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-10-26 Classification: Hydrolase/Hydrolase Inhibitor Ligands: EDO, ZN, PEG, JN7, PO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: EDO, ZN, PEG, JN7, PO4, DMS
![]() |
Crystal Structure Of The Importin-Alpha(44-54)-Importin-Alpha(70-529) Complex
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2001-11-14 Classification: PROTEIN TRANSPORT |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2001-11-14
![]() |
Structure Of Phosphorylated Phenylalanine Hydroxylase
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1999-04-30 Classification: OXIDOREDUCTASE Ligands: FE |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 1999-04-30
Ligands: FE
![]() |
Structure Of Phenylalanine Hydroxylase Dephosphorylated
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 1999-04-30 Classification: OXIDOREDUCTASE Ligands: FE |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 1999-04-30
Ligands: FE
