Search Count: 19
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Bace1 In Complex With (S)-5-(3-Chloro-5-(5-(Prop-1-Yn-1-Yl)Pyridin-3-Yl)Thiophen-2-Yl)-2,5-Dimethyl-1,2,4-Thiadiazinan-3-Iminium 1,1-Dioxide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66J
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Bace1 In Complex With 4-(3-(Furan-2-Carboxamido)Phenyl)-1-Methyl-5-Oxo-4-Phenylimidazolidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: TLA, 66H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: TLA, 66H
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Bace1 In Complex With (R)-N-(3-(3-Amino-2,5-Dimethyl-1,1-Dioxido-5,6-Dihydro-2H-1,2,4-Thiadiazin-5-Yl)-4-Fluorophenyl)-5-Fluoropicolinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66F
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Renin In Complex With (S)-1-(3-Fluoro-5-(((S)-1-Phenylethyl)Carbamoyl)Benzyl)-4-Isopropyl-4-Methyl-6-Oxotetrahydropyrimidin-2(1H)-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-02-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 43T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-25
Ligands: NAG, 43T
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Renin In Complex With (S)-1-(3-(Benzylcarbamoyl)Benzyl)-4-Isopropyl-4-Methyl-6-Oxotetrahydropyrimidin-2(1H)-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-02-18 Classification: Hydrolase/Hydrolase Inhibitor Ligands: NAG, 70X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-18
Ligands: NAG, 70X
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Renin In Complex With (4S)-4-Isopropyl-4-Methyl-6-Oxo-1-(3-(2-Oxo-4-Phenylpyrrolidin-1-Yl)Benzyl)Tetrahydropyrimidin-2(1H)-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-02-18 Classification: Hydrolase/Hydrolase Inhibitor Ligands: NAG, 70Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-18
Ligands: NAG, 70Y
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Structure Of Bace Bound To 2-Imino-3-Methyl-5,5-Diphenylimidazolidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-03-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0KK, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0KK, TLA
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Structure Of Bace Bound To 2-Imino-5-(3'-Methoxy-[1,1'-Biphenyl]-3-Yl)-3-Methyl-5-Phenylimidazolidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2012-03-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0KM, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0KM, TLA
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Structure Of Bace Bound To 2-Imino-3-Methyl-5-Phenyl-5-(3-(Pyridin-3-Yl)Phenyl)Imidazolidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-03-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0KP, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0KP, TLA
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Structure Of Bace Bound To 5-(3-(5-Chloropyridin-3-Yl)Phenyl)-5-Cyclopropyl-2-Imino-3-Methylimidazolidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2012-03-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0KQ, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0KQ, TLA
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Structure Of Bace Bound To (R)-5-Cyclopropyl-2-Imino-3-Methyl-5-(3-(5-(Prop-1-Yn-1-Yl)Pyridin-3-Yl)Phenyl)Imidazolidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2012-03-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0KR, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: 0KR, TLA
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Structure Of Bace Bound To Sch727596
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2008-06-10 Classification: HYDROLASE Ligands: 314, TAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: 314, TAR
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Structure Of Bace Bound To Sch709583
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2008-06-10 Classification: HYDROLASE Ligands: 316, TAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: 316, TAR
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Structure Of Bace Bound To Sch726222
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2008-06-10 Classification: HYDROLASE Ligands: 318, TAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-10
Ligands: 318, TAR
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Structure Of Bace Bound To Sch745966
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2008-03-18 Classification: HYDROLASE Ligands: SC6, TAR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-18
Ligands: SC6, TAR
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Structure Of Bace1 Bound To Sch626485
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-03-11 Classification: HYDROLASE Ligands: CS5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-11
Ligands: CS5
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Structure Of Bace Bound To Sch722924
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2008-03-11 Classification: HYDROLASE Ligands: TAR, CS7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-11
Ligands: TAR, CS7
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Structure Of Bace Bound To Sch735310
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2008-03-11 Classification: HYDROLASE Ligands: TAR, CS9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-11
Ligands: TAR, CS9
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Structure Of Bace Bound To Sch734723
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2008-03-11 Classification: HYDROLASE Ligands: TAR, SC7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-03-11
Ligands: TAR, SC7
