Search Count: 10
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Crystal Structure Of 11B-Hydroxysteroid Dehydrogenase-1 (11B-Hsd1) In Complex With Piperidyl Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-06-16 Classification: OXIDOREDUCTASE Ligands: NAP, A49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-16
Ligands: NAP, A49
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Further Studies With The 2-Amino-1,3-Thiazol-4(5H)-One Class Of 11-Hydroxysteroid Dehydrogenase Type 1 (11-Hsd1) Inhibitors: Reducing Pregnane X Receptor (Pxr) Activity And Exploring Activity In A Monkey Pharmacodynamic Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2008-11-11 Classification: OXIDOREDUCTASE Ligands: NDP, 352 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-11
Ligands: NDP, 352
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase (Hsd1) In Complex With Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-07-22 Classification: OXIDOREDUCTASE Ligands: NAP, D4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-22
Ligands: NAP, D4N
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Crystal Structure Of Human 11-Beta-Hydroxysteroid Dehydrogenase (Hsd1) In Complex With Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-07-01 Classification: OXIDOREDUCTASE Ligands: NAP, D3E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-01
Ligands: NAP, D3E
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The Discovery Of 2-Anilinothiazolones As 11Beta-Hsd1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2008-01-15 Classification: OXIDOREDUCTASE Ligands: ZMG, NDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: ZMG, NDP
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Hiv-1 Protease-Inhibitor Complex
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1999-02-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1IN |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1999-02-23
Ligands: 1IN
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Hiv-1 Protease-Inhibitor Complex
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 1999-02-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1IN |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1999-02-23
Ligands: 1IN
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Hiv-1 Protease-Inhibitor Complex
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 1999-02-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MK1 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1999-02-23
Ligands: MK1
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Hiv-1 Protease-Inhibitor Complex
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1999-02-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3IN |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1999-02-23
Ligands: 3IN
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Hiv-1 Protease-Inhibitor Complex
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1999-02-23 Classification: HYDROLASE/HYDROLASE Ligands: 3IN |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 1999-02-23
Ligands: 3IN
