Search Count: 24
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Crystal Structure Of Mertk Kinase Domain In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2025-10-08 Classification: TRANSFERASE Ligands: A1L6J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-08
Ligands: A1L6J
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Crystal Structure Of Mertk Kinase Domain In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2025-10-08 Classification: TRANSFERASE Ligands: A1L6K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-08
Ligands: A1L6K
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Crystal Structure Of Mertk Kinase Domain In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2025-10-08 Classification: TRANSFERASE Ligands: A1L6L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-08
Ligands: A1L6L
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Crystal Structure Of Jmjd2A Complexed With 3,4-Dihydroxybenzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2022-05-18 Classification: OXIDOREDUCTASE Ligands: DHB, NI, ZN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: DHB, NI, ZN, CL
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Crystal Structure Of Egfr Kinase Domain In Complex With Compound 78
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2019-12-04 Classification: TRANSFERASE/INHIBITOR Ligands: CKO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: CKO
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Crystal Structure Of Egfr Kinase Domain In Complex With Compound 2A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KJQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: KJQ
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Crystal Structure Of Egfr Kinase Domain In Complex With Compound 4B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KJ8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: KJ8
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Crystal Structure Of Egfr Kinase Domain In Complex With Compound 3G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KJR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: KJR
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Crystal Structure Of Egfr Kinase Domain In Complex With Compound 4C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-06-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: KJV
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Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2013-06-05 Classification: TRANSFERASE Ligands: WPH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: WPH
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Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2013-06-05 Classification: TRANSFERASE Ligands: YPH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: YPH
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Novel Aurora Kinase Inhibitors Reveal Mechanisms Of Hurp In Nucleation Of Centrosomal And Kinetochore Microtubules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-06-05 Classification: TRANSFERASE Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-05
Ligands: VX6
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Crystal Structure Of Human Ppar-Gamma Ligand Binding Domain Complex With A Potency Improved Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2011-06-29 Classification: TRANSCRIPTION Ligands: 5BC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-29
Ligands: 5BC
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Crystal Structure Of Aurora A Kinase Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2011-03-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: AKI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-09
Ligands: AKI
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Identification, Sar Studies And X-Ray Cocrystal Analysis Of A Novel Furano-Pyrimidine Aurora Kinase A Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: PFQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: PFQ
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Structure-Based Drug Design Of Novel Aurora Kinase A Inhibitors: Structure Basis For Potency And Specificity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-09-15 Classification: TRANSFERASE Ligands: MMH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-09-15
Ligands: MMH
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Structural Basis For The Structure-Activity Relationships Of Peroxisome Proliferator-Activated Receptor Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2007-08-07 Classification: LIGAND BINDING PROTEIN Ligands: DRY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-07
Ligands: DRY
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Structural Basis For The Structure-Activity Relationships Of Peroxisome Proliferator-Activated Receptor Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2007-08-07 Classification: LIGAND BINDING PROTEIN Ligands: DRD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-07
Ligands: DRD
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Structure-Based Drug Design And Structural Biology Study Of Novel Nonpeptide Inhibitors Of Sars-Cov Main Protease
Organism: Sars coronavirus
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2006-08-29 Classification: HYDROLASE Ligands: D3F |
Organism: Sars coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2006-08-29
Ligands: D3F
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Structure-Based Drug Design And Structural Biology Study Of Novel Nonpeptide Inhibitors Of Sars-Cov Main Protease
Organism: Sars coronavirus
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2006-08-29 Classification: HYDROLASE Ligands: F3F |
Organism: Sars coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2006-08-29
Ligands: F3F
