Search Count: 20
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Bruton'S Tyrosine Kinase In Complex With Covalent Inhibitor Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: UEO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: UEO
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Bruton'S Tyrosine Kinase In Complex With Covalent Inhibitor Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: V72 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: V72
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Bruton'S Tyrosine Kinase In Complex With Covalent Inhibitor Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: V7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: V7I
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Irak4 In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: X1T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: X1T
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Irak4 In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-06-26 Classification: TRANSFERASE/INHIBITOR Ligands: WFQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: WFQ
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Bruton'S Tyrosine Kinase In Complex With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: ZB9, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: ZB9, DMS, PEG
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Bruton'S Tyrosine Kinase In Complex With An Orthosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-03-01 Classification: TRANSFERASE/INHIBITOR Ligands: DMS, Y8C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: DMS, Y8C
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Bruton'S Tyrosine Kinase In Complex With An Orthosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-03-01 Classification: TRANSFERASE/INHIBITOR Ligands: DMS, Y8H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: DMS, Y8H
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Structure Of Compound 34 Bound To Human Phospholipase D2 Catalytic Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2023-01-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CI0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-25
Ligands: CI0
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Bruton'S Tyrosine Kinase In Complex With Compound 45
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B9
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Bruton'S Tyrosine Kinase In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0BG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0BG, DMS
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Bruton'S Tyrosine Kinase In Complex With Compound 65
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0B0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-18
Ligands: 0B0
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Bruton'S Tyrosine Kinase In Complex With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YD7, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: YD7, DMS
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Bruton'S Tyrosine Kinase In Complex With Compound 51
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2022-01-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YDA, DTT, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-12
Ligands: YDA, DTT, ACT
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Bruton'S Tyrosine Kinase In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2020-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DMS, RQS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: DMS, RQS
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Bruton'S Tyrosine Kinase In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DMS, DTT, S5M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: DMS, DTT, S5M
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Bruton'S Tyrosine Kinase In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2020-12-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: S9A, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: S9A, DMS
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Brutons Tyrosine Kinase In Complex With Compound 50.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-06-12 Classification: transferase/transferase inhibitor Ligands: L9S, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: L9S, EDO
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The 1.6 A Crystal Structure Of Human Bruton'S Tyrosine Kinase Bound To A Pyrrolopyrimidine-Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-01-19 Classification: TRANSFERASE Ligands: B43 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: B43
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Structures Of Human Bruton'S Tyrosine Kinase In Active And Inactive Conformations Suggests A Mechanism Of Activation For Tec Family Kinases.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2010-01-19 Classification: TRANSFERASE Ligands: 1N1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: 1N1
