Search Count: 19
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Crystal Structure Of Trim58 Pry-Spry Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2024-01-31 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
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Crystal Structure Of The Trim58 Pry-Spry Domain In Complex With Trim-473
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2024-01-31 Classification: TRANSFERASE Ligands: YCB, MG, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
Ligands: YCB, MG, CL, EDO
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 1: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HJW
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 2 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKE, CHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKE, CHD
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 4 At 2.2A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HKZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HKZ
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Rorcvar2 (Rorgt, 264-499) In Complex With Compound 9 At 2.3A: Identification Of N-Aryl Imidazoles As Potent And Selective Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: HL8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: HL8
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Rorgt (264-518;C455S) In Complex With The Fragment ("Cpd-1") And Rip140 Peptide At 1.80A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EE8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EE8
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Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-2" And Rip140 Peptide At 1.90A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EF5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EF5
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Rorgt (264-518;C455S) In Complex With Inverse Agonist "Cpd-9" And Rip140 Peptide At 1.66A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2018-07-18 Classification: TRANSCRIPTION Ligands: EEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: EEZ
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Discovery Of Cdz173 (Leniolisib), Representing A Structurally Novel Class Of Pi3K Delta-Selective Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-09-20 Classification: TRANSFERASE Ligands: 9NQ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-09-20
Ligands: 9NQ
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: C3S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: C3S
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-06-21 Classification: NUCLEAR PROTEIN Ligands: 99N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 99N
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 98H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 98H
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 98E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 98E
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 444 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 444
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 98N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 98N
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Structural States Of Rorgt: X-Ray Elucidation Of Molecular Mechanisms And Binding Interactions For Natural And Synthetic Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2017-06-21 Classification: SIGNALING PROTEIN Ligands: 8YB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: 8YB
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Crystal Structure Of Pi3K Alpha With Pi3K Delta Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.02 Å Release Date: 2016-09-07 Classification: Transferase/Protein Transport/Inhibitor Ligands: 6CY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: 6CY
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Discovery And Pharmacological Characterization Of Novel Quinazoline-Based Pi3K Delta-Selective Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-08-10 Classification: TRANSFERASE Ligands: 6CY |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 6CY